DOI

The reaction of 3-aryl-N-(aryl)propiolamides with arenes in TfOH at room temperature for 0.5 h led to 4,4-diaryl-3,4-dihydroquinolin-2-(1H)-ones in yields of 44-98%. The obtained dihydroquinolinones were further transformed into the corresponding N-acyl or N-formyl derivatives. For the latter, the superelectrophilic activation of the N-formyl group by TfOH in the reaction with benzene resulted in the formation of N-(diphenylmethyl)-substituted dihydroquinolinones.

Язык оригиналаанглийский
Страницы (с-по)950-956
Число страниц7
ЖурналBeilstein Journal of Organic Chemistry
Том12
DOI
СостояниеОпубликовано - 11 мая 2016

    Предметные области Scopus

  • Органическая химия

ID: 7576360