Research output: Contribution to journal › Article › peer-review
The reaction of 3-aryl-N-(aryl)propiolamides with arenes in TfOH at room temperature for 0.5 h led to 4,4-diaryl-3,4-dihydroquinolin-2-(1H)-ones in yields of 44-98%. The obtained dihydroquinolinones were further transformed into the corresponding N-acyl or N-formyl derivatives. For the latter, the superelectrophilic activation of the N-formyl group by TfOH in the reaction with benzene resulted in the formation of N-(diphenylmethyl)-substituted dihydroquinolinones.
Original language | English |
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Pages (from-to) | 950-956 |
Number of pages | 7 |
Journal | Beilstein Journal of Organic Chemistry |
Volume | 12 |
DOIs | |
State | Published - 11 May 2016 |
ID: 7576360