Research output: Contribution to journal › Article › peer-review
A four-step approach to 2-aryl-2H-tetrazole-5-carboxamides bearing GPCR-focused N-substituted piperazine residues involves ‘SAFE’ diazotransfer onto 1-(piperazin-1-yl)butane-1,3-diones followed by [3+2] cycloaddition of arenediazonium cations at the intermediate ααα-diazo acetamides. The compounds prepared are intended for photoaffinity labeling of aminergic G-protein coupled receptors.
Original language | English |
---|---|
Pages (from-to) | 604-605 |
Number of pages | 2 |
Journal | Mendeleev Communications |
Volume | 32 |
Issue number | 5 |
Early online date | Oct 2022 |
DOIs | |
State | Published - 2022 |
ID: 100361291