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Synthesis of a library of 2-aryl-2H-tetrazole-5-carboxamides for photoaffinity labeling of aminergic G-protein coupled receptors. / Zhukovsky, Daniil; Kanov, Evgeny; Gainetdinov, Raul; Krasavin, Mikhail.

In: Mendeleev Communications , Vol. 32, No. 5, 2022, p. 604-605.

Research output: Contribution to journal › Article › peer-review

Harvard

Zhukovsky, D, Kanov, E, Gainetdinov, R & Krasavin, M 2022, 'Synthesis of a library of 2-aryl-2H-tetrazole-5-carboxamides for photoaffinity labeling of aminergic G-protein coupled receptors', Mendeleev Communications , vol. 32, no. 5, pp. 604-605. https://doi.org/10.1016/j.mencom.2022.09.011

APA

Zhukovsky, D., Kanov, E., Gainetdinov, R., & Krasavin, M. (2022). Synthesis of a library of 2-aryl-2H-tetrazole-5-carboxamides for photoaffinity labeling of aminergic G-protein coupled receptors. Mendeleev Communications , 32(5), 604-605. https://doi.org/10.1016/j.mencom.2022.09.011

Vancouver

Zhukovsky D, Kanov E, Gainetdinov R, Krasavin M. Synthesis of a library of 2-aryl-2H-tetrazole-5-carboxamides for photoaffinity labeling of aminergic G-protein coupled receptors. Mendeleev Communications . 2022;32(5):604-605. https://doi.org/10.1016/j.mencom.2022.09.011

Author

Zhukovsky, Daniil ; Kanov, Evgeny ; Gainetdinov, Raul ; Krasavin, Mikhail. / Synthesis of a library of 2-aryl-2H-tetrazole-5-carboxamides for photoaffinity labeling of aminergic G-protein coupled receptors. In: Mendeleev Communications . 2022 ; Vol. 32, No. 5. pp. 604-605.

BibTeX

@article{2a04e1446f504aa78fd574168a16f52a,
title = "Synthesis of a library of 2-aryl-2H-tetrazole-5-carboxamides for photoaffinity labeling of aminergic G-protein coupled receptors",
abstract = "A four-step approach to 2-aryl-2H-tetrazole-5-carboxamides bearing GPCR-focused N-substituted piperazine residues involves {\textquoteleft}SAFE{\textquoteright} diazotransfer onto 1-(piperazin-1-yl)butane-1,3-diones followed by [3+2] cycloaddition of arenediazonium cations at the intermediate ααα-diazo acetamides. The compounds prepared are intended for photoaffinity labeling of aminergic G-protein coupled receptors.",
keywords = "GPCR privileged ligands, photoaffinity labeling, silver(t) catalysis, tetrazoles, [3+2] cycloaddition, α-diazo acetamides",
author = "Daniil Zhukovsky and Evgeny Kanov and Raul Gainetdinov and Mikhail Krasavin",
note = "Publisher Copyright: {\textcopyright} 2022",
year = "2022",
doi = "10.1016/j.mencom.2022.09.011",
language = "English",
volume = "32",
pages = "604--605",
journal = "Mendeleev Communications",
issn = "0959-9436",
publisher = "Elsevier",
number = "5",

}

RIS

TY - JOUR

T1 - Synthesis of a library of 2-aryl-2H-tetrazole-5-carboxamides for photoaffinity labeling of aminergic G-protein coupled receptors

AU - Zhukovsky, Daniil

AU - Kanov, Evgeny

AU - Gainetdinov, Raul

AU - Krasavin, Mikhail

N1 - Publisher Copyright: © 2022

PY - 2022

Y1 - 2022

N2 - A four-step approach to 2-aryl-2H-tetrazole-5-carboxamides bearing GPCR-focused N-substituted piperazine residues involves ‘SAFE’ diazotransfer onto 1-(piperazin-1-yl)butane-1,3-diones followed by [3+2] cycloaddition of arenediazonium cations at the intermediate ααα-diazo acetamides. The compounds prepared are intended for photoaffinity labeling of aminergic G-protein coupled receptors.

AB - A four-step approach to 2-aryl-2H-tetrazole-5-carboxamides bearing GPCR-focused N-substituted piperazine residues involves ‘SAFE’ diazotransfer onto 1-(piperazin-1-yl)butane-1,3-diones followed by [3+2] cycloaddition of arenediazonium cations at the intermediate ααα-diazo acetamides. The compounds prepared are intended for photoaffinity labeling of aminergic G-protein coupled receptors.

KW - GPCR privileged ligands

KW - photoaffinity labeling

KW - silver(t) catalysis

KW - tetrazoles

KW - [3+2] cycloaddition

KW - α-diazo acetamides

UR - http://www.scopus.com/inward/record.url?scp=85139333311&partnerID=8YFLogxK

UR - https://www.mendeley.com/catalogue/c78a571f-5bc8-34e6-8165-7626a9a4689a/

U2 - 10.1016/j.mencom.2022.09.011

DO - 10.1016/j.mencom.2022.09.011

M3 - Article

AN - SCOPUS:85139333311

VL - 32

SP - 604

EP - 605

JO - Mendeleev Communications

JF - Mendeleev Communications

SN - 0959-9436

IS - 5

ER -

ID: 100361291