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Phosphorylated flavonoids as selective carboxylesterase inhibitors. / Abzianidze, Victoria V. ; Prokofieva, Daria S. ; Beltyukov, Petr P. ; Kuznetsov, Victor A. ; Bogachenkov, Alexander S. ; Rodygin, Konstantin S. .

In: Mendeleev Communications, Vol. 29, No. 1, 02.2019, p. 61-63.

Research output: Contribution to journal › Article › peer-review

Harvard

Abzianidze, VV, Prokofieva, DS, Beltyukov, PP, Kuznetsov, VA, Bogachenkov, AS & Rodygin, KS 2019, 'Phosphorylated flavonoids as selective carboxylesterase inhibitors', Mendeleev Communications, vol. 29, no. 1, pp. 61-63. https://doi.org/10.1016/j.mencom.2019.01.020

APA

Abzianidze, V. V., Prokofieva, D. S., Beltyukov, P. P., Kuznetsov, V. A., Bogachenkov, A. S., & Rodygin, K. S. (2019). Phosphorylated flavonoids as selective carboxylesterase inhibitors. Mendeleev Communications, 29(1), 61-63. https://doi.org/10.1016/j.mencom.2019.01.020

Vancouver

Abzianidze VV, Prokofieva DS, Beltyukov PP, Kuznetsov VA, Bogachenkov AS, Rodygin KS. Phosphorylated flavonoids as selective carboxylesterase inhibitors. Mendeleev Communications. 2019 Feb;29(1):61-63. https://doi.org/10.1016/j.mencom.2019.01.020

Author

Abzianidze, Victoria V. ; Prokofieva, Daria S. ; Beltyukov, Petr P. ; Kuznetsov, Victor A. ; Bogachenkov, Alexander S. ; Rodygin, Konstantin S. . / Phosphorylated flavonoids as selective carboxylesterase inhibitors. In: Mendeleev Communications. 2019 ; Vol. 29, No. 1. pp. 61-63.

BibTeX

@article{2ed5aa640b844c20a6386e60a81d82f5,
title = "Phosphorylated flavonoids as selective carboxylesterase inhibitors",
abstract = "A series of phosphorylated flavonoids has been synthesized and evaluated in vitro for inhibitory activity against carboxylesterase, acetylcholinesterase and butyrylcholinesterase as well as for their cytotoxicity towards human adenocarcinoma A549 and human glioblastoma U251 cell lines. Diethylphosphoryl derivatives of chrysin and 7-hydroxyflavone were found to be the most effective with bimolecular rate constants for carboxylesterase inhibition k i = 2.0 × 10 6 and 5.7 × 10 6 dm 3 mol −1 min −1 , respectively. ",
author = "Abzianidze, {Victoria V.} and Prokofieva, {Daria S.} and Beltyukov, {Petr P.} and Kuznetsov, {Victor A.} and Bogachenkov, {Alexander S.} and Rodygin, {Konstantin S.}",
year = "2019",
month = feb,
doi = "10.1016/j.mencom.2019.01.020",
language = "English",
volume = "29",
pages = "61--63",
journal = "Mendeleev Communications",
issn = "0959-9436",
publisher = "Elsevier",
number = "1",

}

RIS

TY - JOUR

T1 - Phosphorylated flavonoids as selective carboxylesterase inhibitors

AU - Abzianidze, Victoria V.

AU - Prokofieva, Daria S.

AU - Beltyukov, Petr P.

AU - Kuznetsov, Victor A.

AU - Bogachenkov, Alexander S.

AU - Rodygin, Konstantin S.

PY - 2019/2

Y1 - 2019/2

N2 - A series of phosphorylated flavonoids has been synthesized and evaluated in vitro for inhibitory activity against carboxylesterase, acetylcholinesterase and butyrylcholinesterase as well as for their cytotoxicity towards human adenocarcinoma A549 and human glioblastoma U251 cell lines. Diethylphosphoryl derivatives of chrysin and 7-hydroxyflavone were found to be the most effective with bimolecular rate constants for carboxylesterase inhibition k i = 2.0 × 10 6 and 5.7 × 10 6 dm 3 mol −1 min −1 , respectively.

AB - A series of phosphorylated flavonoids has been synthesized and evaluated in vitro for inhibitory activity against carboxylesterase, acetylcholinesterase and butyrylcholinesterase as well as for their cytotoxicity towards human adenocarcinoma A549 and human glioblastoma U251 cell lines. Diethylphosphoryl derivatives of chrysin and 7-hydroxyflavone were found to be the most effective with bimolecular rate constants for carboxylesterase inhibition k i = 2.0 × 10 6 and 5.7 × 10 6 dm 3 mol −1 min −1 , respectively.

UR - http://www.scopus.com/inward/record.url?scp=85061545561&partnerID=8YFLogxK

U2 - 10.1016/j.mencom.2019.01.020

DO - 10.1016/j.mencom.2019.01.020

M3 - Article

VL - 29

SP - 61

EP - 63

JO - Mendeleev Communications

JF - Mendeleev Communications

SN - 0959-9436

IS - 1

ER -

ID: 36903742