Standard

Non-natural 2 : H -azirine-2-carboxylic acids: An expedient synthesis and antimicrobial activity. / Sakharov, Pavel A.; Koronatov, Alexander N.; Khlebnikov, Alexander F.; Novikov, Mikhail S.; Glukharev, Artem G.; Rogacheva, Elizaveta V.; Kraeva, Liudmila A.; Sharoyko, Vladimir V.; Tennikova, Tatiana B.; Rostovskii, Nikolai V.

In: RSC Advances, Vol. 9, No. 65, 2019, p. 37901-37905.

Research output: Contribution to journalArticlepeer-review

Harvard

APA

Vancouver

Author

Sakharov, Pavel A. ; Koronatov, Alexander N. ; Khlebnikov, Alexander F. ; Novikov, Mikhail S. ; Glukharev, Artem G. ; Rogacheva, Elizaveta V. ; Kraeva, Liudmila A. ; Sharoyko, Vladimir V. ; Tennikova, Tatiana B. ; Rostovskii, Nikolai V. / Non-natural 2 : H -azirine-2-carboxylic acids: An expedient synthesis and antimicrobial activity. In: RSC Advances. 2019 ; Vol. 9, No. 65. pp. 37901-37905.

BibTeX

@article{fb4a4ae844dc49ee87b849b70076e8ee,
title = "Non-natural 2: H -azirine-2-carboxylic acids: An expedient synthesis and antimicrobial activity",
abstract = "Non-natural 2H-azirine-2-carboxylic acids were obtained in high yields by FeCl2-catalyzed isomerization of 5-chloroisoxazoles to azirine-2-carbonyl chlorides followed by their hydrolysis. The 3-aryl- and 3-heteroaryl-substituted acids are stable during prolonged storage, exhibit antibacterial activity against ESKAPE pathogens and show a low level of cytotoxicity.",
author = "Sakharov, {Pavel A.} and Koronatov, {Alexander N.} and Khlebnikov, {Alexander F.} and Novikov, {Mikhail S.} and Glukharev, {Artem G.} and Rogacheva, {Elizaveta V.} and Kraeva, {Liudmila A.} and Sharoyko, {Vladimir V.} and Tennikova, {Tatiana B.} and Rostovskii, {Nikolai V.}",
note = "Publisher Copyright: {\textcopyright} 2019 The Royal Society of Chemistry.",
year = "2019",
doi = "10.1039/c9ra09345a",
language = "English",
volume = "9",
pages = "37901--37905",
journal = "RSC Advances",
issn = "2046-2069",
publisher = "Royal Society of Chemistry",
number = "65",

}

RIS

TY - JOUR

T1 - Non-natural 2

T2 - H -azirine-2-carboxylic acids: An expedient synthesis and antimicrobial activity

AU - Sakharov, Pavel A.

AU - Koronatov, Alexander N.

AU - Khlebnikov, Alexander F.

AU - Novikov, Mikhail S.

AU - Glukharev, Artem G.

AU - Rogacheva, Elizaveta V.

AU - Kraeva, Liudmila A.

AU - Sharoyko, Vladimir V.

AU - Tennikova, Tatiana B.

AU - Rostovskii, Nikolai V.

N1 - Publisher Copyright: © 2019 The Royal Society of Chemistry.

PY - 2019

Y1 - 2019

N2 - Non-natural 2H-azirine-2-carboxylic acids were obtained in high yields by FeCl2-catalyzed isomerization of 5-chloroisoxazoles to azirine-2-carbonyl chlorides followed by their hydrolysis. The 3-aryl- and 3-heteroaryl-substituted acids are stable during prolonged storage, exhibit antibacterial activity against ESKAPE pathogens and show a low level of cytotoxicity.

AB - Non-natural 2H-azirine-2-carboxylic acids were obtained in high yields by FeCl2-catalyzed isomerization of 5-chloroisoxazoles to azirine-2-carbonyl chlorides followed by their hydrolysis. The 3-aryl- and 3-heteroaryl-substituted acids are stable during prolonged storage, exhibit antibacterial activity against ESKAPE pathogens and show a low level of cytotoxicity.

UR - http://www.scopus.com/inward/record.url?scp=85075716325&partnerID=8YFLogxK

U2 - 10.1039/c9ra09345a

DO - 10.1039/c9ra09345a

M3 - Article

AN - SCOPUS:85075716325

VL - 9

SP - 37901

EP - 37905

JO - RSC Advances

JF - RSC Advances

SN - 2046-2069

IS - 65

ER -

ID: 99348481