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Fluoroaziridines as novel substrates in the modified Petasis reaction: synthesis of monofluorinated propargyl amines. / Konev, A.S.; Stas, S.; Novikov, M.S.; Khlebnikov, A.F.; Tehrani, K. Abbaspour.

In: Tetrahedron, No. 1, 2008, p. 117-123.

Research output: Contribution to journal › Article

Harvard

Konev, AS, Stas, S, Novikov, MS, Khlebnikov, AF & Tehrani, KA 2008, 'Fluoroaziridines as novel substrates in the modified Petasis reaction: synthesis of monofluorinated propargyl amines', Tetrahedron, no. 1, pp. 117-123. <http://elibrary.ru/item.asp?id=11794221>

APA

Konev, A. S., Stas, S., Novikov, M. S., Khlebnikov, A. F., & Tehrani, K. A. (2008). Fluoroaziridines as novel substrates in the modified Petasis reaction: synthesis of monofluorinated propargyl amines. Tetrahedron, (1), 117-123. http://elibrary.ru/item.asp?id=11794221

Vancouver

Konev AS, Stas S, Novikov MS, Khlebnikov AF, Tehrani KA. Fluoroaziridines as novel substrates in the modified Petasis reaction: synthesis of monofluorinated propargyl amines. Tetrahedron. 2008;(1):117-123.

Author

Konev, A.S. ; Stas, S. ; Novikov, M.S. ; Khlebnikov, A.F. ; Tehrani, K. Abbaspour. / Fluoroaziridines as novel substrates in the modified Petasis reaction: synthesis of monofluorinated propargyl amines. In: Tetrahedron. 2008 ; No. 1. pp. 117-123.

BibTeX

@article{c51775aa3038471a86cd7f5a6c4f6701,
title = "Fluoroaziridines as novel substrates in the modified Petasis reaction: synthesis of monofluorinated propargyl amines",
abstract = "Reaction of 2-fluoroaziridines with potassium alkynyltrifluoroborates in the presence of BF3·OEt2 leads to fluorinated propargyl amines in moderate to good yields. The reaction proceeds as an in situ isomerization of 2-fluoroaziridines to α-fluorinated imines, followed by the reaction of the imine with alkynyldifluoroborane, which is generated in situ from the potassium alkynyltrifluoroborates and BF3·OEt2. {\textcopyright} 2007 Elsevier Ltd. All rights reserved.",
author = "A.S. Konev and S. Stas and M.S. Novikov and A.F. Khlebnikov and Tehrani, {K. Abbaspour}",
year = "2008",
language = "English",
pages = "117--123",
journal = "Tetrahedron",
issn = "0040-4020",
publisher = "Elsevier",
number = "1",

}

RIS

TY - JOUR

T1 - Fluoroaziridines as novel substrates in the modified Petasis reaction: synthesis of monofluorinated propargyl amines

AU - Konev, A.S.

AU - Stas, S.

AU - Novikov, M.S.

AU - Khlebnikov, A.F.

AU - Tehrani, K. Abbaspour

PY - 2008

Y1 - 2008

N2 - Reaction of 2-fluoroaziridines with potassium alkynyltrifluoroborates in the presence of BF3·OEt2 leads to fluorinated propargyl amines in moderate to good yields. The reaction proceeds as an in situ isomerization of 2-fluoroaziridines to α-fluorinated imines, followed by the reaction of the imine with alkynyldifluoroborane, which is generated in situ from the potassium alkynyltrifluoroborates and BF3·OEt2. © 2007 Elsevier Ltd. All rights reserved.

AB - Reaction of 2-fluoroaziridines with potassium alkynyltrifluoroborates in the presence of BF3·OEt2 leads to fluorinated propargyl amines in moderate to good yields. The reaction proceeds as an in situ isomerization of 2-fluoroaziridines to α-fluorinated imines, followed by the reaction of the imine with alkynyldifluoroborane, which is generated in situ from the potassium alkynyltrifluoroborates and BF3·OEt2. © 2007 Elsevier Ltd. All rights reserved.

M3 - Article

SP - 117

EP - 123

JO - Tetrahedron

JF - Tetrahedron

SN - 0040-4020

IS - 1

ER -

ID: 5009863