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1,3,5-Triazinanes as Formaldimine Surrogates in the Ugi Reaction. / Golubev, Pavel; Guranova, Natalia; Krasavin, Mikhail.

In: European Journal of Organic Chemistry, Vol. 2020, No. 29, 09.08.2020, p. 4517-4520.

Research output: Contribution to journal › Article › peer-review

Harvard

Golubev, P, Guranova, N & Krasavin, M 2020, '1,3,5-Triazinanes as Formaldimine Surrogates in the Ugi Reaction', European Journal of Organic Chemistry, vol. 2020, no. 29, pp. 4517-4520. https://doi.org/10.1002/ejoc.202000569

APA

Golubev, P., Guranova, N., & Krasavin, M. (2020). 1,3,5-Triazinanes as Formaldimine Surrogates in the Ugi Reaction. European Journal of Organic Chemistry, 2020(29), 4517-4520. https://doi.org/10.1002/ejoc.202000569

Vancouver

Golubev P, Guranova N, Krasavin M. 1,3,5-Triazinanes as Formaldimine Surrogates in the Ugi Reaction. European Journal of Organic Chemistry. 2020 Aug 9;2020(29):4517-4520. https://doi.org/10.1002/ejoc.202000569

Author

Golubev, Pavel ; Guranova, Natalia ; Krasavin, Mikhail. / 1,3,5-Triazinanes as Formaldimine Surrogates in the Ugi Reaction. In: European Journal of Organic Chemistry. 2020 ; Vol. 2020, No. 29. pp. 4517-4520.

BibTeX

@article{d117891472564c97bfc2ecc6895ed48a,
title = "1,3,5-Triazinanes as Formaldimine Surrogates in the Ugi Reaction",
abstract = "In the present study, a new synthetic strategy towards N-acylated glycinamides was developed by the use of 1,3,5-triazinanes as formaldimine surrogates in the Ugi reaction. The targeted products were obtained in a combinatorial, diversity-oriented fashion in good yields. Further modifications allowed us to adapt this procedure for the one-pot two-step syntheses of a local anesthetic druglidocaine and several unsymmetrically substituted diketopiperazines.",
keywords = "1,3,5-Triazinanes, Molecular diversity, Multicomponent reactions, Synthetic methods, Ugi reaction",
author = "Pavel Golubev and Natalia Guranova and Mikhail Krasavin",
year = "2020",
month = aug,
day = "9",
doi = "10.1002/ejoc.202000569",
language = "English",
volume = "2020",
pages = "4517--4520",
journal = "European Journal of Organic Chemistry",
issn = "1434-193X",
publisher = "Wiley-Blackwell",
number = "29",

}

RIS

TY - JOUR

T1 - 1,3,5-Triazinanes as Formaldimine Surrogates in the Ugi Reaction

AU - Golubev, Pavel

AU - Guranova, Natalia

AU - Krasavin, Mikhail

PY - 2020/8/9

Y1 - 2020/8/9

N2 - In the present study, a new synthetic strategy towards N-acylated glycinamides was developed by the use of 1,3,5-triazinanes as formaldimine surrogates in the Ugi reaction. The targeted products were obtained in a combinatorial, diversity-oriented fashion in good yields. Further modifications allowed us to adapt this procedure for the one-pot two-step syntheses of a local anesthetic druglidocaine and several unsymmetrically substituted diketopiperazines.

AB - In the present study, a new synthetic strategy towards N-acylated glycinamides was developed by the use of 1,3,5-triazinanes as formaldimine surrogates in the Ugi reaction. The targeted products were obtained in a combinatorial, diversity-oriented fashion in good yields. Further modifications allowed us to adapt this procedure for the one-pot two-step syntheses of a local anesthetic druglidocaine and several unsymmetrically substituted diketopiperazines.

KW - 1,3,5-Triazinanes

KW - Molecular diversity

KW - Multicomponent reactions

KW - Synthetic methods

KW - Ugi reaction

UR - http://www.scopus.com/inward/record.url?scp=85088103523&partnerID=8YFLogxK

U2 - 10.1002/ejoc.202000569

DO - 10.1002/ejoc.202000569

M3 - Article

AN - SCOPUS:85088103523

VL - 2020

SP - 4517

EP - 4520

JO - European Journal of Organic Chemistry

JF - European Journal of Organic Chemistry

SN - 1434-193X

IS - 29

ER -

ID: 61393926