Panel docking of small-molecule libraries - Prospects to improve efficiency of lead compound discovery

Sarnpitak, P., Mujumdar, P., Taylor, P., Cross, M., Coster, M. J., Gorse, A. D., Krasavin, M. & Hofmann, A., 1 Nov 2015, In: Biotechnology Advances. 33, 6, p. 941-947 7 p.

Research output: Contribution to journal › Review article › peer-review

Atom-economical construction of tetracyclic [1,4]oxazepines involving intramolecular arylation of a 2-imidazoline moiety

Karamysheva, K., Reutskaya, E., Sapegin, A., Dorogov, M. & Krasavin, M., 7 Oct 2015, In: Tetrahedron Letters. 56, 41, p. 5632-5636 5 p.

Research output: Contribution to journal › Article › peer-review

A convenient preparation of diversely substituted fused 2-amino- and 2-alkylthionicotinonitriles under microwave irradiation

Krasavin, M., Sapegin, A. & Dorogov, M., 2015, In: Tetrahedron Letters. 56, 1, p. 56-60

Research output: Contribution to journal › Article

An improved kilogram-scale preparation of atorvastatin calcium

Novozhilov, Y. V., Dorogov, M. V., Blumina, M. V., Smirnov, A. V. & Krasavin, M., 2015, In: Chemistry Central Journal. 9

Research output: Contribution to journal › Article › peer-review

Biologically active compounds based on the privileged 2-imidazoline scaffold: the world beyond adrenergic/imidazoline receptor modulators

Krasavin, M., 2015, In: European Journal of Medicinal Chemistry. 97, p. 525-537

Research output: Contribution to journal › Review article › peer-review

Discovery of 2-[1-(4,4-Difluorocyclohexyl)piperidin-4-yl]-6-fluoro-3-oxo-2,3-dihydro-1H-isoindole-4-carboxamide (NMS-P118): A Potent, Orally Available, and Highly Selective PARP-1 Inhibitor for Cancer Therapy

Papeo, G., Posteri, H., Borghi, D., Busel, A. A., Caprera, F., Casale, E., Ciomei, M., Cirla, A., Corti, E., D'Anello, M., Fasolini, M., Forte, B., Galvani, A., Isacchi, A., Khvat, A., Krasavin, M. Y., Lupi, R., Orsini, P., Perego, R., Pesenti, E. & 9 others, Pezzetta, D., Rainoldi, S., Riccardi-Sirtori, F., Scolaro, A., Sola, F., Zuccotto, F., Felder, E. R., Donati, D. & Montagnoli, A., 2015, In: Journal of Medicinal Chemistry. 17, p. 6875-6898

Research output: Contribution to journal › Article

Efficient Use of 1,2-Dihaloazine Synthons in Transition-Metal-Free Preparation of Doverse Heterocycle-Fused 1,4-Oxazepines

Sapegin, A. V., Kalinin, S. A., Smirnov, A. V., Dorogov, M. V. & Krasavin, M., 2015, In: European Journal of Organic Chemistry. 2015, 6, p. 1333-1340

Research output: Contribution to journal › Article › peer-review

Facile Pd-catalyzed amination of imidazolin-1-yl chloroazines under microwave irradiation: toward a new kinase-inhibitory chemotype

Mujumdar, P., Sarnpitak, P., Shetnev, A., Dorogov, M. & Krasavin, M., 2015, In: Tetrahedron Letters. 56, p. 2827-2831

Research output: Contribution to journal › Article

New Heterocyclic Product Space for the Castagnoli-Cushman Three-Component Reaction

Dar'In, D., Bakulina, O., Chizhova, M. & Krasavin, M., 2015, In: Organic Letters. p. 3930-3933

Research output: Contribution to journal › Article

Pd-catalyzed amination of imidazolin-1-yl azines: toward a new kinase-inhibitory chemotype.

Красавин, М. Ю., 2015, In: Tetrahedron Letters. 56, p. 2827-2831

Research output: Contribution to journal › Article › peer-review