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  1. 2023

  2. Synthesis of novel glutarimide ligands for the E3 ligase substrate receptor Cereblon (CRBN): Investigation of their binding mode and antiproliferative effects against myeloma cell lines

    Krasavin, M., Adamchik, M., Bubyrev, A., Heim, C., Maiwald, S., Zhukovsky, D., Zhmurov, P., Bunev, A. & Hartmann, M. D., 15 Jan 2023, In: European Journal of Medicinal Chemistry. 246, 114990.

    Research output: Contribution to journal › Article › peer-review

  3. Synthesis of novel glutarimide derivatives via the Michael addition of (hetero)aromatic thiols: pronounced effect of sulfur oxidation on cytotoxicity towards multiple myeloma cell lines

    Адамчик, М. А., Бубырев, А. И., Жуковский, Д. Д., Жмуров, П. А., Бунев, А. С. & Красавин, М. Ю., 1 Jan 2023, In: Mendeleev Communications. 33, 1, p. 67-69 3 p.

    Research output: Contribution to journal › Article › peer-review

  4. 2022

  5. Diversely substituted sulfamides for fragment-based drug discovery of carbonic anhydrase inhibitors: synthesis and inhibitory profile

    Sharonova, T., Zhmurov, P., Kalinin, S., Nocentini, A., Angeli, A., Ferraroni, M., Korsakov, M., Supuran, C. T. & Krasavin, M., 16 Mar 2022, In: Journal of Enzyme Inhibition and Medicinal Chemistry. 37, 1, p. 857-865 9 p.

    Research output: Contribution to journal › Article › peer-review

  6. 2021

  7. 1-Oxo-3,4-dihydroisoquinoline-4-carboxamides as novel druglike inhibitors of poly(ADP-ribose) polymerase (PARP) with favourable ADME characteristics

    Safrygin, A., Zhmurov, P., Dar’in, D., Silonov, S., Kasatkina, M., Zonis, Y., Gureev, M. & Krasavin, M., 1 Jan 2021, In: Journal of Enzyme Inhibition and Medicinal Chemistry. 36, 1, p. 1968-1983 16 p.

    Research output: Contribution to journal › Article › peer-review

  8. Three-component Castagnoli-Cushman reaction with ammonium acetate delivers 2-unsubstituted isoquinol-1-ones as potent inhibitors of poly(ADP-ribose) polymerase (PARP)

    Safrygin, A., Zhmurov, P., Dar’in, D., Silonov, S., Kasatkina, M., Zonis, Y., Gureev, M. & Krasavin, M., 2021, In: Journal of Enzyme Inhibition and Medicinal Chemistry. 36, 1, p. 1916-1921 6 p.

    Research output: Contribution to journal › Article › peer-review

  9. 2020

  10. α-Diazoacetamides in Sc(OTf) 3 -Catalyzed Tiffeneau-Demjanov Ring Expansion: Application towards the Synthesis of Rare Bicyclic Pyrazoles

    Chuprun, S., Dar'In, D., Kantin, G., Zhmurov, P. & Krasavin, M., 3 Mar 2020, In: Synlett. 31, 4, p. 373-377 5 p., st-2019-b0609-l.

    Research output: Contribution to journal › Article › peer-review

  11. Sulfocoumarins as dual inhibitors of human carbonic anhydrase isoforms IX/XII and of human thioredoxin reductase

    Krasavin, M., Žalubovskis, R., Grandāne, A., Domračeva, I., Zhmurov, P. & Supuran, C. T., 1 Jan 2020, In: Journal of Enzyme Inhibition and Medicinal Chemistry. 35, 1, p. 506-510 5 p.

    Research output: Contribution to journal › Article › peer-review

  12. One-pot preparation of methyl 2-diazo-3-oxopropionates comprising an aqueous ‘sulfonyl-azide-free’ (SAFE) diazo transfer step

    Zhmurov, P. A., Dar'in, D. V., Bakulina, O. Y. & Krasavin, M., 2020, In: Mendeleev Communications . 30, 3, p. 311-312 2 p.

    Research output: Contribution to journal › Article › peer-review

  13. Taking diazo transfer to water: alpha-diazo carbonyl compounds from in situ generated mesyl azide

    Shevalev, R. M., Zhmurov, P. A., Dar'in, D. V. & Krasavin, M., 2020, In: Mendeleev Communications . 30, 3, p. 372-373 2 p.

    Research output: Contribution to journal › Article › peer-review

  14. 2018

  15. A Novel Entry to 3,4,5-Trisubstituted 2-Pyrrolidones from Isoxazoline-N-oxides

    Zhmurov, P. A., Ushakov, P. Y., Novikov, R. A., Sukhorukov, A. Y. & Ioffe, S. L., 1 Jan 2018, In: Synlett. 29, 14, p. 1871-1874 4 p.

    Research output: Contribution to journal › Article › peer-review

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