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  1. 2021

  2. Exploration of the nitrogen heterocyclic periphery around the core of the advanced FFA1 agonist fasiglifam (TAK-875)

    Lukin, A., Bakholdina, A., Zhurilo, N., Onopchenko, O., Zhuravel, E., Zozulya, S., Gureev, M., Safrygin, A. & Krasavin, M., Apr 2021, In: Archiv der Pharmazie. 354, 4, 16 p., 2000275.

    Research output: Contribution to journal › Article › peer-review

  3. 1-Oxo-3,4-dihydroisoquinoline-4-carboxamides as novel druglike inhibitors of poly(ADP-ribose) polymerase (PARP) with favourable ADME characteristics

    Safrygin, A., Zhmurov, P., Dar’in, D., Silonov, S., Kasatkina, M., Zonis, Y., Gureev, M. & Krasavin, M., 1 Jan 2021, In: Journal of Enzyme Inhibition and Medicinal Chemistry. 36, 1, p. 1968-1983 16 p.

    Research output: Contribution to journal › Article › peer-review

  4. Three-component Castagnoli-Cushman reaction with ammonium acetate delivers 2-unsubstituted isoquinol-1-ones as potent inhibitors of poly(ADP-ribose) polymerase (PARP)

    Safrygin, A., Zhmurov, P., Dar’in, D., Silonov, S., Kasatkina, M., Zonis, Y., Gureev, M. & Krasavin, M., 2021, In: Journal of Enzyme Inhibition and Medicinal Chemistry. 36, 1, p. 1916-1921 6 p.

    Research output: Contribution to journal › Article › peer-review

  5. 2020

  6. Synthesis of spirocyclic tetrahydroisoquinolines (spiroTHIQs) via the Castagnoli-Cushman reaction

    Safrygin, A., Dar'in, D., Bakulina, O. & Krasavin, M., 15 Oct 2020, In: Tetrahedron Letters. 61, 42, 3 p., 152408.

    Research output: Contribution to journal › Article › peer-review

  7. Three-Component Reaction of Homophthalic Anhydride with Carbonyl Compounds and Ammonium Acetate: New Developments

    Safrygin, A., Bakulina, O., Dar'In, D. & Krasavin, M., 4 Aug 2020, In: Synthesis (Germany). 52, 15, p. 2190-2195 6 p.

    Research output: Contribution to journal › Article › peer-review

  8. 2019

  9. α-Diazo-β-oxosulfones as Partners in the Wolff 1,2,3-Triazole Synthesis and the Wolff Rearrangement in the Presence of Aromatic Amines

    Safrygin, A., Dar'in, D., Kantin, G. & Krasavin, M., 7 Aug 2019, In: European Journal of Organic Chemistry. 2019, 29, p. 4721-4724 4 p.

    Research output: Contribution to journal › Article › peer-review

  10. Erratum to “Zn(OTf) 2 -catalyzed, microwave-promoted synthesis of 2-substituted 5-methyloxazoles from propargylic amides” [Tetrahedron Lett. 60 (2019) 777–779](S0040403919301182)(10.1016/j.tetlet.2019.02.011)

    Safrygin, A., Dar'in, D., Lukin, A., Bakholdina, A., Sapegin, A. & Krasavin, M., 16 May 2019, In: Tetrahedron Letters. 60, 20, p. 1397-1398 2 p.

    Research output: Contribution to journal › Comment/debate › peer-review

  11. Zn(OTf)2-catalyzed, microwave-promoted synthesis of 2-substituted 5-methyloxazoles from propargylic amides

    Safrygin, A., Dar'in, D., Lukin, A., Bakholdina, A., Sapegin, A. & Krasavin, M., 14 Mar 2019, In: Tetrahedron Letters. 60, 11, p. 777-779 3 p.

    Research output: Contribution to journal › Article › peer-review

  12. 2018

  13. Efficient Conversion of Tertiary Propargylamides into Imidazoles via Hydroamination-Cyclization

    Safrygin, A., Krivosheyeva, E., Dar'in, D. & Krasavin, M., 1 Aug 2018, In: Synthesis (Germany). 50, 15, p. 3048-3058 11 p., ss-2018-z0257-op.

    Research output: Contribution to journal › Article › peer-review

ID: 6810669