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Diversity-oriented synthesis of N,N-dimethylamino-substituted azoles employing TBTU. / Lukin, Alexey; Kalinchenkova, Natalya; Vedekhina, Tatiana; Zhurilo, Nikolay; Krasavin, Mikhail.

в: Tetrahedron Letters, Том 59, № 28, 11.07.2018, стр. 2732-2735.

Результаты исследований: Научные публикации в периодических изданиях › статья › Рецензирование

Harvard

Lukin, A, Kalinchenkova, N, Vedekhina, T, Zhurilo, N & Krasavin, M 2018, 'Diversity-oriented synthesis of N,N-dimethylamino-substituted azoles employing TBTU', Tetrahedron Letters, Том. 59, № 28, стр. 2732-2735. https://doi.org/10.1016/j.tetlet.2018.05.075

APA

Lukin, A., Kalinchenkova, N., Vedekhina, T., Zhurilo, N., & Krasavin, M. (2018). Diversity-oriented synthesis of N,N-dimethylamino-substituted azoles employing TBTU. Tetrahedron Letters, 59(28), 2732-2735. https://doi.org/10.1016/j.tetlet.2018.05.075

Vancouver

Lukin A, Kalinchenkova N, Vedekhina T, Zhurilo N, Krasavin M. Diversity-oriented synthesis of N,N-dimethylamino-substituted azoles employing TBTU. Tetrahedron Letters. 2018 Июль 11;59(28):2732-2735. https://doi.org/10.1016/j.tetlet.2018.05.075

Author

Lukin, Alexey ; Kalinchenkova, Natalya ; Vedekhina, Tatiana ; Zhurilo, Nikolay ; Krasavin, Mikhail. / Diversity-oriented synthesis of N,N-dimethylamino-substituted azoles employing TBTU. в: Tetrahedron Letters. 2018 ; Том 59, № 28. стр. 2732-2735.

BibTeX

@article{00bc4af3ad7f4f558ade7f3b4d83d50a,
title = "Diversity-oriented synthesis of N,N-dimethylamino-substituted azoles employing TBTU",
abstract = "A convenient, diversity-oriented approach for the transformation of readily available amidoximes, o-hydroxyarylamines, acyl hydrazines, carboximidohydrazides and thiohydrazides into their respective N,N-dimethylamino-substituted azoles is described. The method is particularly suitable for array chemistry application as it employs a stable, solid reagent TBTU.",
keywords = "Acylation, Azoles, Dimethylamino group, Diversity-oriented synthesis, Fragment-based drug discovery, Guanidine formation, REAGENT, LEAD DISCOVERY, DRUG DISCOVERY, DERIVATIVES, SALTS",
author = "Alexey Lukin and Natalya Kalinchenkova and Tatiana Vedekhina and Nikolay Zhurilo and Mikhail Krasavin",
year = "2018",
month = jul,
day = "11",
doi = "10.1016/j.tetlet.2018.05.075",
language = "English",
volume = "59",
pages = "2732--2735",
journal = "Tetrahedron Letters",
issn = "0040-4039",
publisher = "Elsevier",
number = "28",

}

RIS

TY - JOUR

T1 - Diversity-oriented synthesis of N,N-dimethylamino-substituted azoles employing TBTU

AU - Lukin, Alexey

AU - Kalinchenkova, Natalya

AU - Vedekhina, Tatiana

AU - Zhurilo, Nikolay

AU - Krasavin, Mikhail

PY - 2018/7/11

Y1 - 2018/7/11

N2 - A convenient, diversity-oriented approach for the transformation of readily available amidoximes, o-hydroxyarylamines, acyl hydrazines, carboximidohydrazides and thiohydrazides into their respective N,N-dimethylamino-substituted azoles is described. The method is particularly suitable for array chemistry application as it employs a stable, solid reagent TBTU.

AB - A convenient, diversity-oriented approach for the transformation of readily available amidoximes, o-hydroxyarylamines, acyl hydrazines, carboximidohydrazides and thiohydrazides into their respective N,N-dimethylamino-substituted azoles is described. The method is particularly suitable for array chemistry application as it employs a stable, solid reagent TBTU.

KW - Acylation

KW - Azoles

KW - Dimethylamino group

KW - Diversity-oriented synthesis

KW - Fragment-based drug discovery

KW - Guanidine formation

KW - REAGENT

KW - LEAD DISCOVERY

KW - DRUG DISCOVERY

KW - DERIVATIVES

KW - SALTS

UR - http://www.scopus.com/inward/record.url?scp=85048327311&partnerID=8YFLogxK

U2 - 10.1016/j.tetlet.2018.05.075

DO - 10.1016/j.tetlet.2018.05.075

M3 - Article

AN - SCOPUS:85048327311

VL - 59

SP - 2732

EP - 2735

JO - Tetrahedron Letters

JF - Tetrahedron Letters

SN - 0040-4039

IS - 28

ER -

ID: 34632504