Research output: Contribution to journal › Article › peer-review
Synthesis of benzannelated sultams by intramolecular Pd-catalyzed arylation of tertiary sulfonamides. / Соколов, Виктор Владимирович; Рассадин, Валентин Анатольевич.
In: Beilstein Journal of Organic Chemistry, Vol. 13, 10.3762/bjoc.13.187, 12.09.2017, p. 1932-1939.Research output: Contribution to journal › Article › peer-review
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TY - JOUR
T1 - Synthesis of benzannelated sultams by intramolecular Pd-catalyzed arylation of tertiary sulfonamides
AU - Соколов, Виктор Владимирович
AU - Рассадин, Валентин Анатольевич
PY - 2017/9/12
Y1 - 2017/9/12
N2 - A new and efficient approach to five- and six-membered benzannelated sultams by intramolecular C-arylation of tertiary1-(methoxycarbonyl)methanesulfonamides under palladium catalysis is described. In case of the α-toluenesulfonamide derivative,an unexpected formation of a 2,3-diarylindole was observed under the same conditions.
AB - A new and efficient approach to five- and six-membered benzannelated sultams by intramolecular C-arylation of tertiary1-(methoxycarbonyl)methanesulfonamides under palladium catalysis is described. In case of the α-toluenesulfonamide derivative,an unexpected formation of a 2,3-diarylindole was observed under the same conditions.
KW - arylation; fused-ring systems; indole formation; palladium catalysis; sultams
U2 - 10.3762/bjoc.13.187
DO - 10.3762/bjoc.13.187
M3 - Article
VL - 13
SP - 1932
EP - 1939
JO - Beilstein Journal of Organic Chemistry
JF - Beilstein Journal of Organic Chemistry
SN - 1860-5397
M1 - 10.3762/bjoc.13.187
ER -
ID: 9328650