The interaction of the ethyl ester or pyrrolidide of 3, 3-diaminoacrylic acid with aromatic and heteroaromatic nitriles containing a labile halogen atom in the ortho position, leads to the formation of products of its substitution by the α-carbon atom of the diaminoacrylic acid derivative. The compounds obtained are cyclized smoothly into fused diaminoazines.

Original languageEnglish
Pages (from-to)436-441
Number of pages6
JournalChemistry of Heterocyclic Compounds
Volume48
Issue number3
DOIs
StatePublished - 2012

    Scopus subject areas

  • Organic Chemistry

    Research areas

  • 3,3-diaminoacrylic acid derivatives, Fused diaminoazines, O-haloarenecarbonitriles

ID: 5482048