N-amination of unsymmetrically substituted pyrimidines. Synthesis of isomeric N-aminopyrimidones

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Magnetic Resonance Research Centre
Department of Organic Chemistry

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DOI

https://doi.org/10.1023/A:1023716424186
Final published version

M. B. Bodyagin
A. Yu Ivanov
K. Wurst
J. G. Schantl
P. S. Lobanov
A. A. Potekhin

N-Amination of 6-amino-2-methyl-4-pyrimidone with O-(mesitylenesulfonyl)hydroxylamine leads to the 3-amino derivative. The isomeric 1,6-diamino-2-methyl-4-pyrimidone was obtained by the N-amination of the O-benzoyl derivative of the initial pyrimidone and removal of the benzoyl protection.

Original language	English
Pages (from-to)	195-199
Number of pages	5
Journal	Chemistry of Heterocyclic Compounds
Volume	39
Issue number	2
DOIs	https://doi.org/10.1023/A:1023716424186
State	Published - 1 Feb 2003

Scopus subject areas

Organic Chemistry

Research areas

4-pyrimidones, N-amination, O-(mesitylenesulfonyl)hydroxylamine

ID: 36153505