Research output: Contribution to journal › Article › peer-review
A Route to Benzo-Annelated δ-Sultams through Michael Cyclization. / Соколов, Виктор Владимирович; Рассадин, Валентин Анатольевич; Grosheva, Daria S.
In: European Journal of Organic Chemistry, Vol. 6, No. 6, 2015, p. 1355-1363.Research output: Contribution to journal › Article › peer-review
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TY - JOUR
T1 - A Route to Benzo-Annelated δ-Sultams through Michael Cyclization
AU - Соколов, Виктор Владимирович
AU - Рассадин, Валентин Анатольевич
AU - Grosheva, Daria S.
PY - 2015
Y1 - 2015
N2 - A new approach to benzo-annelated δ-sultams containing anaryl–nitrogen bond is described. The method, which involvesthe intramolecular Michael cyclization of tert-butyl ortho-[N-(methoxycarbonylmethyl)sulfonylamino]cinnamates, allows the synthesis of secondary sultams as well as their tertiaryanalogues and bridged tricyclic derivatives efficiently anddiastereoselectively.
AB - A new approach to benzo-annelated δ-sultams containing anaryl–nitrogen bond is described. The method, which involvesthe intramolecular Michael cyclization of tert-butyl ortho-[N-(methoxycarbonylmethyl)sulfonylamino]cinnamates, allows the synthesis of secondary sultams as well as their tertiaryanalogues and bridged tricyclic derivatives efficiently anddiastereoselectively.
KW - Heterocycles / Sultams / Fused-ring systems / Michael addition / Cyclization
U2 - 10.1002/ejoc.201403416
DO - 10.1002/ejoc.201403416
M3 - Article
VL - 6
SP - 1355
EP - 1363
JO - European Journal of Organic Chemistry
JF - European Journal of Organic Chemistry
SN - 1434-193X
IS - 6
ER -
ID: 3927987