Mixed carboxylic-sulfonic anhydride in reaction with imines: A straightforward route to water-soluble β-lactams via a Staudinger-type reaction

Bakulina, O., Dar'in, D. & Krasavin, M., 1 Jan 2018, In: Organic and Biomolecular Chemistry. 16, 21, p. 3989-3998 10 p.

Research output: Contribution to journal › Article › peer-review

Cyclic Hydroxamic Acid Analogues of Bacterial Siderophores as Iron-Complexing Agents prepared through the Castagnoli–Cushman Reaction of Unprotected Oximes

Bakulina, O., Bannykh, A., Dar'in, D. & Krasavin, M., 14 Dec 2017, In: Chemistry - A European Journal. 23, 70, p. 17667-17673 7 p.

Research output: Contribution to journal › Article › peer-review

Skeletal Diversity in Combinatorial Fashion: A New Format for the Castagnoli-Cushman Reaction

Lepikhina, A., Dar'In, D., Bakulina, O., Chupakhin, E. & Krasavin, M., 13 Nov 2017, In: ACS Combinatorial Science. 19, 11, p. 702-707 6 p.

Research output: Contribution to journal › Article › peer-review

Lucky Switcheroo: Dramatic Potency and Selectivity Improvement of Imidazoline Inhibitors of Human Carbonic Anhydrase VII

Kalinin, S., Kopylov, S., Tuccinardi, T., Sapegin, A., Dar'In, D., Angeli, A., Supuran, C. T. & Krasavin, M., 12 Oct 2017, In: ACS Medicinal Chemistry Letters. 8, 10, p. 1105-1109 5 p.

Research output: Contribution to journal › Article › peer-review

1,3-Oxazole-based selective picomolar inhibitors of cytosolic human carbonic anhydrase II alleviate ocular hypertension in rabbits: Potency is supported by X-ray crystallography of two leads

Ferraroni, M., Lucarini, L., Masini, E., Korsakov, M., Scozzafava, A., Supuran, C. T. & Krasavin, M., 1 Sep 2017, In: Bioorganic and Medicinal Chemistry. 25, 17, p. 4560-4565 6 p.

Research output: Contribution to journal › Article › peer-review

A speedy route to sterically encumbered, benzene-fused derivatives of privileged, naturally occurring hexahydropyrrolo[1,2-b]isoquinoline

Bakulina, O., Ivanov, A., Suslonov, V., Darin, D. & Krasavin, M., 18 Jul 2017, In: Beilstein Journal of Organic Chemistry. 13, p. 1413-1424 12 p.

Research output: Contribution to journal › Article › peer-review

Sterically Constrained and Encumbered: An Approach to the Naturally Occurring Peptidomimetic Tetrahydropyrazino[1,2-a]indole-1,4-dione Core

Golubev, P. & Krasavin, M., 3 Apr 2017, In: European Journal of Organic Chemistry. 2017, 13, p. 1740-1744 5 p.

Research output: Contribution to journal › Article › peer-review

Spontaneous formation of tricyclic lactones following the Castagnoli–Cushman reaction

Usmanova, L., Bakulina, O., Dar’in, D. & Krasavin, M., 1 Apr 2017, In: Chemistry of Heterocyclic Compounds. 53, 4, p. 474-479 6 p.

Research output: Contribution to journal › Article › peer-review

Discovery and Preclinical Characterization of 3-((4-(4-Chlorophenyl)-7-fluoroquinoline-3-yl)sulfonyl)benzonitrile, a Novel Non-acetylenic Metabotropic Glutamate Receptor 5 (mGluR5) Negative Allosteric Modulator for Psychiatric Indications

Galambos, J., Bielik, A., Krasavin, M., Orgován, Z., Domány, G., Nógrádi, K., Wágner, G., Balogh, G. T., Béni, Z., Kóti, J., Szakács, Z., Bobok, A., Kolok, S., Mikó-Bakk, M. L., Vastag, M., Sághy, K., Laszy, J., Halász, A. S., Balázs, O., Gál, K. & 3 others, Greiner, I., Szombathelyi, Z. & Keserű, G. M., 23 Mar 2017, In: Journal of Medicinal Chemistry. 60, 6, p. 2470-2484 15 p.

Research output: Contribution to journal › Article › peer-review

N-(Hetero)aryl-2-imidazolines: An emerging privileged motif for contemporary drug design

Krasavin, M., 1 Mar 2017, In: Chemistry of Heterocyclic Compounds. 53, 3, p. 240-255 16 p.

Research output: Contribution to journal › Review article › peer-review