1. 2023
  2. Diazo Tetramic Acids Provide Access to Natural-Like Spirocyclic Δ α,β - Butenolides through Rh(II)-Catalyzed O−H Insertion/Base-Promoted Cyclization

    Дарьин, Д. В., Кантин, Г. П., Глушакова, Д. В., Шаройко, В. В. & Красавин, М. Ю., 5 Jan 2023, (E-pub ahead of print) In: Journal of Organic Chemistry.

    Research output: Contribution to journalArticlepeer-review

  3. Synthesis and Antibacterial Evaluation of Ciprofloxacin Congeners with Spirocyclic Amine Periphery

    Lukin, A., Komarova, K., Vinogradova, L., Rogacheva, E., Kraeva, L. & Krasavin, M., 4 Jan 2023, In: International Journal of Molecular Sciences. 24, 2, 954.

    Research output: Contribution to journalArticlepeer-review

  4. Periphery exploration around 2,6-diazaspiro[3.4]octane core identifies a potent nitrofuran antitubercular lead

    Lukin, A., Yablonsky, P., Komarova, K., Vinogradova, L., Dogonadze, M., Vinogradova, T., Казанцев, А. С. & Красавин, М. Ю., 2023, In: Molecules (Basel, Switzerland). 28, 6, 15 p., 2529.

    Research output: Contribution to journalArticlepeer-review

  5. 2022
  6. 5-(Sulfamoyl)thien-2-yl 1,3-oxazole inhibitors of carbonic anhydrase II with hydrophilic periphery

    Kalinin, S., Kovalenko, A., Valtari, A., Nocentini, A., Gureev, M., Urtti, A., Korsakov, M., Supuran, C. T. & Krasavin, M., 31 Dec 2022, In: Journal of Enzyme Inhibition and Medicinal Chemistry. 37, 1, p. 1005-1011 7 p.

    Research output: Contribution to journalArticlepeer-review

  7. Replacing the phthalimide core in thalidomide with benzotriazole

    Krasavin, M., Bubyrev, A., Kazantsev, A., Heim, C., Maiwald, S., Zhukovsky, D., Dar’in, D., Hartmann, M. D. & Bunev, A., 31 Dec 2022, In: Journal of Enzyme Inhibition and Medicinal Chemistry. 37, 1, p. 527-530 4 p.

    Research output: Contribution to journalArticlepeer-review

  8. A novel bis-triazole scaffold accessed via two tandem [3 + 2] cycloaddition events including an uncatalyzed, room temperature azide–alkyne click reaction

    Malkova, K., Bubyrev, A., Krivovicheva, V., Dar’in, D., Bunev, A. & Krasavin, M., Dec 2022, In: Beilstein Journal of Organic Chemistry. 18, p. 1636-1641

    Research output: Contribution to journalArticlepeer-review

  9. Metal-free synthetic approaches to 1,5-disubstituted 1,2,3-triazoles

    Malkova, K., Bubyrev, A., Balalaie, S., Dar'in, D. & Krasavin, M., Dec 2022, In: Tetrahedron Letters. 112, p. 154228

    Research output: Contribution to journalArticlepeer-review

  10. Synthetic Exploration of Novel Sulfamoyl Cyanide N-Oxides in Heterocycle Synthesis

    Krivovicheva, V., Bubyrev, A., Kalinin, S., Dar'in, D. & Krasavin, M., Dec 2022, In: European Journal of Organic Chemistry. 46, e202201162.

    Research output: Contribution to journalArticlepeer-review

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