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    Author

    Михаил Юрьевич Красавин
2019
Tetrazoles
Silver Nitrate
Cycloaddition
Nitrates
Silver
4 Citations (Scopus)

1,2,4-Oxadiazole/2-Imidazoline Hybrids: Multi-target-directed Compounds for the Treatment of Infectious Diseases and Cancer

Shetnev, A., Baykov, S., Kalinin, S., Belova, A., Sharoyko, V., Rozhkov, A., Zelenkov, L., Tarasenko, M., Sadykov, E., Korsakov, M. & Krasavin, M., 1 Apr 2019, In : International Journal of Molecular Sciences. 20, 7, p. 1699 10 p., 1699.

Research output

Oxadiazoles
infectious diseases
Bacilli
Amides
Scaffolds
Oxazoles
Nitriles
Azides
Cycloaddition
Cycloaddition Reaction
8 Citations (Scopus)
Azides
Scaffolds
Substrates
1 Citation (Scopus)
Open Access
2 Citations (Scopus)
Piperidines
Nitrofurans
Multidrug-Resistant Tuberculosis
Mycobacterium tuberculosis
Retinal Pigments
Ring opening polymerization
quinoline
Zinc
polymerization
zinc

BOB.1 controls memory B-cell fate in the germinal center reaction

Levels, M. J., Fehres, C. M., van Baarsen, L. G. M., van Uden, N. O. P., Germar, K., O'Toole, T. G., Blijdorp, I. C. J., Semmelink, J. F., Doorenspleet, M. E., Bakker, A. Q., Krasavin, M., Tomilin, A., Brouard, S., Spits, H., Baeten, D. L. P. & Yeremenko, N. G., Jul 2019, In : Journal of Autoimmunity. 101, p. 131-144

Research output

1 Citation (Scopus)
Oxidative Coupling
Sulfhydryl Compounds
Thioredoxin Reductase 1
Acids
Disulfides
3 Citations (Scopus)

Effect of chiral polyhydrochromenes on cannabinoid system

Li-Zhulanov, N. S., Il’ina, I. V., Chicca, A., Schenker, P., Patrusheva, O. S., Nazimova, E. V., Korchagina, D. V., Krasavin, M., Volcho, K. P. & Salakhutdinov, N. F., 1 Jan 2019, In : Medicinal Chemistry Research.

Research output

Cannabinoids
Endocannabinoids
Cannabinoid Receptor CB2
Cannabinoid Receptor CB1
Bromine
Open Access
Hydroxamic Acids
Hydroxylamine
format
Iron
Siderophores
Open Access
Selenocysteine
Thioredoxin-Disulfide Reductase
Acids
Palladium
Hydrolysis
1 Citation (Scopus)
Carbonic Anhydrases
Sulfonamides
Cytotoxicity
Glioma
Hydrogen

Highly hydrophilic 1,3-oxazol-5-yl benzenesulfonamide inhibitors of carbonic anhydrase II for reduction of glaucoma-related intraocular pressure

Kalinin, S., Valtari, A., Ruponen, M., Toropainen, E., Kovalenko, A., Nocentini, A., Gureev, M., Dar'in, D., Urtti, A., Supuran, C. T. & Krasavin, M., 1 Jan 2019, In : Bioorganic and Medicinal Chemistry. 115086.

Research output

dorzolamide
Carbonic Anhydrase II
Ophthalmic Solutions
Intraocular Pressure
Glaucoma

Inhibition of Neutrophil Elastase and Cathepsin G As a New Approach to the Treatment of Psoriasis: From Fundamental Biology to Development of New Target-Specific Drugs

Krasavin, M. Y., Gureev, M. A., Garabadzhiu, A. V., Pashkin, A. Y., Zhukov, A. S., Khairutdinov, V. R., Samtsov, A. V. & Shvets, V. I., 2019, In : Doklady Biochemistry and Biophysics. 487, 1, p. 272-276

Research output

Cathepsin G
Leukocyte Elastase
Molecular modeling
Pancreatic Elastase
Serine Proteases
Modular construction
Metal ions
Metals
Ions
Fluorescence
2 Citations (Scopus)
Nevirapine
Crystallization
adducts
Stabilization
stabilization
2 Citations (Scopus)
Imidazolines
Endonucleases
Orthomyxoviridae
Viruses
Human Influenza
2 Citations (Scopus)
Thioredoxin Reductase 1
Lead compounds
Thioredoxins
Videodisks
Amides
1 Citation (Scopus)
Potash
Azides
Ketones
Purification
Esters
3 Citations (Scopus)
Cells
Membranes
Cell Line
Protein Isoforms
Lead compounds
3 Citations (Scopus)
Cyclic Ethers
Cycloaddition
Carbon Monoxide
Decomposition
Scaffolds
1 Citation (Scopus)
Amines
insertion
Aniline Compounds
amines
Sulfonamides

Spirocyclic motifs in natural products

Chupakhin, E., Babich, O., Prosekov, A., Asyakina, L. & Krasavin, M., 17 Nov 2019, In : Molecules. 24, 22, 37 p., 4165.

Research output

Open Access
Biological Products
products
Drug Discovery
voids
emerging
4 Citations (Scopus)

Synthesis of various arylated trifluoromethyl substituted indanes and indenes, and study of their biological activity

Iakovenko, R. O., Chicca, A., Nieri, D., Reynoso-Moreno, I., Gertsch, J., Krasavin, M. & Vasilyev, A. V., Feb 2019, In : Tetrahedron. 75, 5, p. 624-632

Research output

Indenes
Bearings (structural)
Monoacylglycerol Lipases
Endocannabinoids
Cyclization
2 Citations (Scopus)
Imidazoles
Indoles
Amides
Carbon
Atoms
3 Citations (Scopus)
Microwaves
Amides
Microwave irradiation
Toluene
Metals

Zn(OTf)2-catalyzed arenehydrazination of protected propargylamines leading to 3-amidoindoles

Vedekhina, T., Lukin, A., Rogacheva, E., Kraeva, L. & Krasavin, M., 1 Jan 2019, (Accepted/In press) In : Tetrahedron Letters. 151430.

Research output

Bearings (structural)
Nitrogen
Catalysts
Pathogens
Screening
1 Citation (Scopus)
Lactams
Transition metals
Imines
Discrete Fourier transforms
Bearings (structural)
Cycloaddition Reaction
Cyanides
5-hydroxymethylfurfural