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  • 2020
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Author

  • Михаил Юрьевич Красавин
1 Citation (Scopus)

1,2,4-Oxadiazole/2-Imidazoline Hybrids: Multi-target-directed Compounds for the Treatment of Infectious Diseases and Cancer

Shetnev, A., Baykov, S., Kalinin, S., Belova, A., Sharoyko, V., Rozhkov, A., Zelenkov, L., Tarasenko, M., Sadykov, E., Korsakov, M. & Krasavin, M., 1 Apr 2019, In : International Journal of Molecular Sciences. 20, 7, p. 1699 10 p., 1699.

Research output

4 Citations (Scopus)
5 Citations (Scopus)
2 Citations (Scopus)

7-Acylamino-3H-1,2-benzoxathiepine 2,2-dioxides as new isoform-selective carbonic anhydrase IX and XII inhibitors

Pustenko, A., Nocentini, A., Balašova, A., Krasavin, M., Žalubovskis, R. & Supuran, C. T., 21 Feb 2020, In : Journal of Enzyme Inhibition and Medicinal Chemistry. 35, 1, p. 650-656 7 p.

Research output

Open Access
2 Citations (Scopus)
2 Citations (Scopus)
9 Citations (Scopus)
8 Citations (Scopus)

Aldazines in the Castagnoli-Cushman Reaction

Mikheyev, A., Kantin, G. & Krasavin, M., 17 May 2018, In : Synthesis (Germany). 50, 10, p. 2076-2086 11 p.

Research output

1 Citation (Scopus)

Aryl derivatives of 3H-1,2-benzoxathiepine 2,2-dioxide as carbonic anhydrase inhibitors

Pustenko, A., Nocentini, A., Balašova, A., Alafeefy, A., Krasavin, M., Žalubovskis, R. & Supuran, C. T., 1 Jan 2020, In : Journal of Enzyme Inhibition and Medicinal Chemistry. 35, 1, p. 245-254

Research output

Open Access
3 Citations (Scopus)
13 Citations (Scopus)
2 Citations (Scopus)
Open Access
2 Citations (Scopus)
4 Citations (Scopus)
1 Citation (Scopus)

BOB.1 controls memory B-cell fate in the germinal center reaction

Levels, M. J., Fehres, C. M., van Baarsen, L. G. M., van Uden, N. O. P., Germar, K., O'Toole, T. G., Blijdorp, I. C. J., Semmelink, J. F., Doorenspleet, M. E., Bakker, A. Q., Krasavin, M., Tomilin, A., Brouard, S., Spits, H., Baeten, D. L. P. & Yeremenko, N. G., Jul 2019, In : Journal of Autoimmunity. 101, p. 131-144

Research output

Open Access
1 Citation (Scopus)

Conjugation of a 5-nitrofuran-2-oyl moiety to aminoalkylimidazoles produces non-toxic nitrofurans that are efficacious in vitro and in vivo against multidrug-resistant Mycobacterium tuberculosis

Krasavin, M., Lukin, A., Vedekhina, T., Manicheva, O., Dogonadze, M., Vinogradova, T., Zabolotnykh, N., Rogacheva, E., Kraeva, L. & Yablonsky, P., 5 Sep 2018, In : European Journal of Medicinal Chemistry. 157, p. 1115-1126 12 p.

Research output

2 Citations (Scopus)

Continued SAR exploration of 1,2,4-thiadiazole-containing scaffolds in the design of free fatty acid receptor 1 (GPR40) agonists

Krasavin, M., Lukin, A., Bakholdina, A., Zhurilo, N., Onopchenko, O., Borysko, P., Zozulya, S., Moore, D. & Tikhonova, I. G., 1 Jan 2017, In : European Journal of Medicinal Chemistry. 140, p. 229-238 10 p.

Research output

5 Citations (Scopus)
5 Citations (Scopus)

Design, in silico prioritization and biological profiling of apoptosis-inducing lactams amenable by the Castagnoli-Cushman reaction

Krasavin, M., Gureyev, M. A., Dar'in, D., Bakulina, O., Chizhova, M., Lepikhina, A., Novikova, D., Grigoreva, T., Ivanov, G., Zhumagalieva, A., Garabadzhiu, A. V. & Tribulovich, V. G., 15 May 2018, In : Bioorganic and Medicinal Chemistry. 26, 9, p. 2651-2673 23 p.

Research output

2 Citations (Scopus)
2 Citations (Scopus)

Discovery and Preclinical Characterization of 3-((4-(4-Chlorophenyl)-7-fluoroquinoline-3-yl)sulfonyl)benzonitrile, a Novel Non-acetylenic Metabotropic Glutamate Receptor 5 (mGluR5) Negative Allosteric Modulator for Psychiatric Indications

Galambos, J., Bielik, A., Krasavin, M., Orgován, Z., Domány, G., Nógrádi, K., Wágner, G., Balogh, G. T., Béni, Z., Kóti, J., Szakács, Z., Bobok, A., Kolok, S., Mikó-Bakk, M. L., Vastag, M., Sághy, K., Laszy, J., Halász, A. S., Balázs, O., Gál, K. & 3 others, Greiner, I., Szombathelyi, Z. & Keserű, G. M., 23 Mar 2017, In : Journal of Medicinal Chemistry. 60, 6, p. 2470-2484 15 p.

Research output

11 Citations (Scopus)

Discovery of 4-amino-3-arylsulfoquinolines, a novel non-acetylenic chemotype of metabotropic glutamate 5 (mGlu5) receptor negative allosteric modulators

Galambos, J., Bielik, A., Wágner, G., Domány, G., Kóti, J., Béni, Z., Szigetvári, Á., Sánta, Z., Orgován, Z., Bobok, A., Kiss, B., Mikó-Bakk, M. L., Vastag, M., Sághy, K., Krasavin, M., Gál, K., Greiner, I., Szombathelyi, Z. & Keserű, G. M., 1 Jan 2017, In : European Journal of Medicinal Chemistry. 133, p. 240-254 15 p.

Research output

4 Citations (Scopus)

Discovery of polar spirocyclic orally bioavailable urea inhibitors of soluble epoxide hydrolase

Lukin, A., Kramer, J., Hartmann, M., Weizel, L., Hernandez-Olmos, V., Falahati, K., Burghardt, I., Kalinchenkova, N., Bagnyukova, D., Zhurilo, N., Rautio, J., Forsberg, M., Ihalainen, J., Auriola, S., Leppänen, J., Konstantinov, I., Pogoryelov, D., Proschak, E., Dar'in, D. & Krasavin, M., 1 Oct 2018, In : Bioorganic Chemistry. 80, p. 655-667 13 p.

Research output

6 Citations (Scopus)
3 Citations (Scopus)

Diversity-oriented synthesis of N,N-dimethylamino-substituted azoles employing TBTU

Lukin, A., Kalinchenkova, N., Vedekhina, T., Zhurilo, N. & Krasavin, M., 11 Jul 2018, In : Tetrahedron Letters. 59, 28, p. 2732-2735 4 p.

Research output

1 Citation (Scopus)

Effect of chiral polyhydrochromenes on cannabinoid system

Li-Zhulanov, N. S., Il’ina, I. V., Chicca, A., Schenker, P., Patrusheva, O. S., Nazimova, E. V., Korchagina, D. V., Krasavin, M., Volcho, K. P. & Salakhutdinov, N. F., Apr 2019, In : Medicinal Chemistry Research. 28, 4, p. 450-464

Research output

3 Citations (Scopus)

Efficient Conversion of Tertiary Propargylamides into Imidazoles via Hydroamination-Cyclization

Safrygin, A., Krivosheyeva, E., Dar'in, D. & Krasavin, M., 1 Aug 2018, In : Synthesis (Germany). 50, 15, p. 3048-3058 11 p., ss-2018-z0257-op.

Research output

7 Citations (Scopus)

Efficient cyclodehydration of dicarboxylic acids with oxalyl chloride

Kantin, G., Chupakhin, E., Dar'in, D. & Krasavin, M., 1 Jan 2017, In : Tetrahedron Letters. 58, 32, p. 3160-3163 4 p.

Research output

10 Citations (Scopus)
2 Citations (Scopus)
3 Citations (Scopus)

Exploring bulky natural and natural-like periphery in the design of p-(benzyloxy)phenylpropionic acid agonists of free fatty acid receptor 1 (GPR40)

Kuranov, S. O., Luzina, O. A., Onopchenko, O., Pishel, I., Zozulya, S., Gureev, M., Salakhutdinov, N. F. & Krasavin, M., Jun 2020, In : Bioorganic Chemistry. 99, 103830.

Research output

3 Citations (Scopus)