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Publication Year

  • 2020
  • 2019
  • 2018
  • 2017
  • 2016

Author

  • Михаил Юрьевич Красавин
5 Citations (Scopus)
3 Citations (Scopus)

Free fatty acid receptor 1 (GPR40) agonists containing spirocyclic periphery inspired by LY2881835

Krasavin, M., Lukin, A., Bagnyukova, D., Zhurilo, N., Zahanich, I., Zozulya, S., Ihalainen, J., Forsberg, M. M., Lehtonen, M., Rautio, J., Moore, D. & Tikhonova, I. G., 1 Nov 2016, In : Bioorganic and Medicinal Chemistry. 24, 21, p. 5481-5494 14 p.

Research output

11 Citations (Scopus)

Gram-scale synthesis of a novel core building block for the new GPR40 agonist design

Lukin, A., Bagnyukova, D., Zhurilo, N. & Krasavin, M., 1 Aug 2016, In : Letters in Organic Chemistry. 13, 7, p. 491-495 5 p.

Research output

2 Citations (Scopus)

Isoform-selective inhibitory profile of 2-imidazoline-substituted benzenesulfonamides against a panel of human carbonic anhydrases.

Supuran, C. T., Kalinin, S., Tanç, M., Sarnpitak, P., Mujumdar, P., Poulsen, SA. & Krasavin, M., 2016, In : Journal of Enzyme Inhibition and Medicinal Chemistry. 31 (Suppl. 1), p. 197-202

Research output

21 Citations (Scopus)

Library of diversely substituted 2-(quinolin-4-yl)imidazolines delivers novel non-cytotoxic antitubercular leads

Krasavin, M., Mujumdar, P., Parchinsky, V., Vinogradova, T., Manicheva, O. & Dogonadze, M., 1 Nov 2016, In : Journal of Enzyme Inhibition and Medicinal Chemistry. 31, 6, p. 1146-1155 10 p.

Research output

8 Citations (Scopus)
11 Citations (Scopus)

New antimycobacterial leads from multicomponent hydrazino-ugi reaction

Lakontseva, E., Karapetian, R. & Krasavin, M., 1 Mar 2016, In : Medicinal Chemistry. 12, 2, p. 191-199 9 p.

Research output

2 Citations (Scopus)
2 Citations (Scopus)
7 Citations (Scopus)
2017
5 Citations (Scopus)
1 Citation (Scopus)

Continued SAR exploration of 1,2,4-thiadiazole-containing scaffolds in the design of free fatty acid receptor 1 (GPR40) agonists

Krasavin, M., Lukin, A., Bakholdina, A., Zhurilo, N., Onopchenko, O., Borysko, P., Zozulya, S., Moore, D. & Tikhonova, I. G., 1 Jan 2017, In : European Journal of Medicinal Chemistry. 140, p. 229-238 10 p.

Research output

5 Citations (Scopus)

Discovery and Preclinical Characterization of 3-((4-(4-Chlorophenyl)-7-fluoroquinoline-3-yl)sulfonyl)benzonitrile, a Novel Non-acetylenic Metabotropic Glutamate Receptor 5 (mGluR5) Negative Allosteric Modulator for Psychiatric Indications

Galambos, J., Bielik, A., Krasavin, M., Orgován, Z., Domány, G., Nógrádi, K., Wágner, G., Balogh, G. T., Béni, Z., Kóti, J., Szakács, Z., Bobok, A., Kolok, S., Mikó-Bakk, M. L., Vastag, M., Sághy, K., Laszy, J., Halász, A. S., Balázs, O., Gál, K. & 3 others, Greiner, I., Szombathelyi, Z. & Keserű, G. M., 23 Mar 2017, In : Journal of Medicinal Chemistry. 60, 6, p. 2470-2484 15 p.

Research output

12 Citations (Scopus)

Discovery of 4-amino-3-arylsulfoquinolines, a novel non-acetylenic chemotype of metabotropic glutamate 5 (mGlu5) receptor negative allosteric modulators

Galambos, J., Bielik, A., Wágner, G., Domány, G., Kóti, J., Béni, Z., Szigetvári, Á., Sánta, Z., Orgován, Z., Bobok, A., Kiss, B., Mikó-Bakk, M. L., Vastag, M., Sághy, K., Krasavin, M., Gál, K., Greiner, I., Szombathelyi, Z. & Keserű, G. M., 1 Jan 2017, In : European Journal of Medicinal Chemistry. 133, p. 240-254 15 p.

Research output

4 Citations (Scopus)

Efficient cyclodehydration of dicarboxylic acids with oxalyl chloride

Kantin, G., Chupakhin, E., Dar'in, D. & Krasavin, M., 1 Jan 2017, In : Tetrahedron Letters. 58, 32, p. 3160-3163 4 p.

Research output

11 Citations (Scopus)

Fluorescent (pyrazolyl acetoxime)Zn-II complexes: Synthetic, structural, and photophysical studies

Bolotin, D. S., Il'in, M. V., Kolesnikov, I. E., Suslonov, V. V., Novozhilov, Y., Ronzhina, O., Krasavin, M., Boyarskiy, V. P., Koen, R. & Roodt, A., 30 Jan 2017, In : Inorganica Chimica Acta. 455, p. 9-14 6 p.

Research output

3 Citations (Scopus)

Human carbonic anhydrase inhibitory profile of mono- and bis-sulfonamides synthesized via a direct sulfochlorination of 3- and 4-(hetero)arylisoxazol-5-amine scaffolds

Krasavin, M., Korsakov, M., Zvonaryova, Z., Semyonychev, E., Tuccinardi, T., Kalinin, S., Tanç, M. & Supuran, C. T., 1 Jan 2017, In : Bioorganic and Medicinal Chemistry. 25, 6, p. 1914-1925 12 p.

Research output

11 Citations (Scopus)
7 Citations (Scopus)
1 Citation (Scopus)
7 Citations (Scopus)

New nitrofurans amenable by isocyanide multicomponent chemistry are active against multidrug-resistant and poly-resistant Mycobacterium tuberculosis

Krasavin, M., Parchinsky, V., Kantin, G., Manicheva, O., Dogonadze, M., Vinogradova, T., Karge, B. & Brönstrup, M., 1 Jan 2017, In : Bioorganic and Medicinal Chemistry. 25, 6, p. 1867-1874 8 p.

Research output

12 Citations (Scopus)

Novel FFA1 (GPR40) agonists containing spirocyclic periphery: polar azine periphery as a driver of potency

Krasavin, M., Lukin, A., Bagnyukova, D., Zhurilo, N., Zahanich, I. & Zozulya, S., 1 Jan 2017, In : Journal of Enzyme Inhibition and Medicinal Chemistry. 32, 1, p. 29-36 8 p.

Research output

3 Citations (Scopus)

Polar aromatic periphery increases agonist potency of spirocyclic free fatty acid receptor (GPR40) agonists inspired by LY2881835

Krasavin, M., Lukin, A., Bagnyukova, D., Zhurilo, N., Golovanov, A., Zozulya, S., Zahanich, I., Moore, D. & Tikhonova, I. G., 1 Jan 2017, In : European Journal of Medicinal Chemistry. 127, p. 357-368 12 p.

Research output

3 Citations (Scopus)
14 Citations (Scopus)

Short Approach to Pyrrolopyrazino-, Pyrrolodiazepino-Isoindoles and their Benzo Analogues via the IMDAF Reaction

Zubkov, F. I., Orlova, D. N., Zaytsev, V. P., Voronov, A. A., Nikitina, E. V., Khrustalev, V. N., Novikov, R. A., Krasavin, M. & Varlamov, A. V., 2017, In : Current Organic Synthesis. 14, 5, p. 733-746 14 p.

Research output

12 Citations (Scopus)
9 Citations (Scopus)
16 Citations (Scopus)

Synthesis, structure and properties of N-aminosaccharine – a selective inhibitor of human carbonic anhydrase I

Kuznetsov, M. A., Shestakov, A. N., Zibinsky, M., Krasavin, M., Supuran, C. T., Kalinin, S. & Tanç, M., 2017, In : Tetrahedron Letters. 58, 2, p. 172-174

Research output

2 Citations (Scopus)
2018
2 Citations (Scopus)