Find Research Outputs

Search in all content

Filters for Research Output

Search concepts
Selected filters

Publication Year

  • 2020
  • 2019
  • 2017
  • 2016

Author

  • Михаил Юрьевич Красавин

Free fatty acid receptor 1 (GPR40) agonists containing spirocyclic periphery inspired by LY2881835

Krasavin, M., Lukin, A., Bagnyukova, D., Zhurilo, N., Zahanich, I., Zozulya, S., Ihalainen, J., Forsberg, M. M., Lehtonen, M., Rautio, J., Moore, D. & Tikhonova, I. G., 1 Nov 2016, In : Bioorganic and Medicinal Chemistry. 24, 21, p. 5481-5494 14 p.

Research output

11 Citations (Scopus)
2017
9 Citations (Scopus)
2017

Synthesis, structure and properties of N-aminosaccharine – a selective inhibitor of human carbonic anhydrase I

Kuznetsov, M. A., Shestakov, A. N., Zibinsky, M., Krasavin, M., Supuran, C. T., Kalinin, S. & Tanç, M., 2017, In : Tetrahedron Letters. 58, 2, p. 172-174

Research output

2 Citations (Scopus)

Novel FFA1 (GPR40) agonists containing spirocyclic periphery: polar azine periphery as a driver of potency

Krasavin, M., Lukin, A., Bagnyukova, D., Zhurilo, N., Zahanich, I. & Zozulya, S., 1 Jan 2017, In : Journal of Enzyme Inhibition and Medicinal Chemistry. 32, 1, p. 29-36 8 p.

Research output

3 Citations (Scopus)

New nitrofurans amenable by isocyanide multicomponent chemistry are active against multidrug-resistant and poly-resistant Mycobacterium tuberculosis

Krasavin, M., Parchinsky, V., Kantin, G., Manicheva, O., Dogonadze, M., Vinogradova, T., Karge, B. & Brönstrup, M., 1 Jan 2017, In : Bioorganic and Medicinal Chemistry. 25, 6, p. 1867-1874 8 p.

Research output

12 Citations (Scopus)
2020
2017

Discovery of 4-amino-3-arylsulfoquinolines, a novel non-acetylenic chemotype of metabotropic glutamate 5 (mGlu5) receptor negative allosteric modulators

Galambos, J., Bielik, A., Wágner, G., Domány, G., Kóti, J., Béni, Z., Szigetvári, Á., Sánta, Z., Orgován, Z., Bobok, A., Kiss, B., Mikó-Bakk, M. L., Vastag, M., Sághy, K., Krasavin, M., Gál, K., Greiner, I., Szombathelyi, Z. & Keserű, G. M., 1 Jan 2017, In : European Journal of Medicinal Chemistry. 133, p. 240-254 15 p.

Research output

4 Citations (Scopus)

Continued SAR exploration of 1,2,4-thiadiazole-containing scaffolds in the design of free fatty acid receptor 1 (GPR40) agonists

Krasavin, M., Lukin, A., Bakholdina, A., Zhurilo, N., Onopchenko, O., Borysko, P., Zozulya, S., Moore, D. & Tikhonova, I. G., 1 Jan 2017, In : European Journal of Medicinal Chemistry. 140, p. 229-238 10 p.

Research output

5 Citations (Scopus)
2019
Open Access
6 Citations (Scopus)
2017

Discovery and Preclinical Characterization of 3-((4-(4-Chlorophenyl)-7-fluoroquinoline-3-yl)sulfonyl)benzonitrile, a Novel Non-acetylenic Metabotropic Glutamate Receptor 5 (mGluR5) Negative Allosteric Modulator for Psychiatric Indications

Galambos, J., Bielik, A., Krasavin, M., Orgován, Z., Domány, G., Nógrádi, K., Wágner, G., Balogh, G. T., Béni, Z., Kóti, J., Szakács, Z., Bobok, A., Kolok, S., Mikó-Bakk, M. L., Vastag, M., Sághy, K., Laszy, J., Halász, A. S., Balázs, O., Gál, K. & 3 others, Greiner, I., Szombathelyi, Z. & Keserű, G. M., 23 Mar 2017, In : Journal of Medicinal Chemistry. 60, 6, p. 2470-2484 15 p.

Research output

12 Citations (Scopus)
2019
9 Citations (Scopus)
21 Citations (Scopus)
2017
9 Citations (Scopus)
2019
5 Citations (Scopus)
2020
2019
2019
4 Citations (Scopus)
2020
1 Citation (Scopus)
2017
7 Citations (Scopus)
2019
3 Citations (Scopus)
2020
1 Citation (Scopus)
Open Access
2019

Inhibition of Neutrophil Elastase and Cathepsin G As a New Approach to the Treatment of Psoriasis: From Fundamental Biology to Development of New Target-Specific Drugs

Krasavin, M. Y., Gureev, M. A., Garabadzhiu, A. V., Pashkin, A. Y., Zhukov, A. S., Khairutdinov, V. R., Samtsov, A. V. & Shvets, V. I., 2019, In : Doklady Biochemistry and Biophysics. 487, 1, p. 272-276

Research output

2017

Fluorescent (pyrazolyl acetoxime)Zn-II complexes: Synthetic, structural, and photophysical studies

Bolotin, D. S., Il'in, M. V., Kolesnikov, I. E., Suslonov, V. V., Novozhilov, Y., Ronzhina, O., Krasavin, M., Boyarskiy, V. P., Koen, R. & Roodt, A., 30 Jan 2017, In : Inorganica Chimica Acta. 455, p. 9-14 6 p.

Research output

3 Citations (Scopus)
2020
2019
2 Citations (Scopus)
2019
3 Citations (Scopus)
2016
7 Citations (Scopus)
5 Citations (Scopus)

Gram-scale synthesis of a novel core building block for the new GPR40 agonist design

Lukin, A., Bagnyukova, D., Zhurilo, N. & Krasavin, M., 1 Aug 2016, In : Letters in Organic Chemistry. 13, 7, p. 491-495 5 p.

Research output

2 Citations (Scopus)

New antimycobacterial leads from multicomponent hydrazino-ugi reaction

Lakontseva, E., Karapetian, R. & Krasavin, M., 1 Mar 2016, In : Medicinal Chemistry. 12, 2, p. 191-199 9 p.

Research output

2 Citations (Scopus)
2017
7 Citations (Scopus)