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Publication Year

  • 2020
  • 2018
  • 2017
  • 2016

Author

  • Михаил Юрьевич Красавин

Free fatty acid receptor 1 (GPR40) agonists containing spirocyclic periphery inspired by LY2881835

Krasavin, M., Lukin, A., Bagnyukova, D., Zhurilo, N., Zahanich, I., Zozulya, S., Ihalainen, J., Forsberg, M. M., Lehtonen, M., Rautio, J., Moore, D. & Tikhonova, I. G., 1 Nov 2016, In : Bioorganic and Medicinal Chemistry. 24, 21, p. 5481-5494 14 p.

Research output

11 Citations (Scopus)
2018

Diversity-oriented synthesis of N,N-dimethylamino-substituted azoles employing TBTU

Lukin, A., Kalinchenkova, N., Vedekhina, T., Zhurilo, N. & Krasavin, M., 11 Jul 2018, In : Tetrahedron Letters. 59, 28, p. 2732-2735 4 p.

Research output

3 Citations (Scopus)
2017
9 Citations (Scopus)
2018
9 Citations (Scopus)
2017

Synthesis, structure and properties of N-aminosaccharine – a selective inhibitor of human carbonic anhydrase I

Kuznetsov, M. A., Shestakov, A. N., Zibinsky, M., Krasavin, M., Supuran, C. T., Kalinin, S. & Tanç, M., 2017, In : Tetrahedron Letters. 58, 2, p. 172-174

Research output

2 Citations (Scopus)

Novel FFA1 (GPR40) agonists containing spirocyclic periphery: polar azine periphery as a driver of potency

Krasavin, M., Lukin, A., Bagnyukova, D., Zhurilo, N., Zahanich, I. & Zozulya, S., 1 Jan 2017, In : Journal of Enzyme Inhibition and Medicinal Chemistry. 32, 1, p. 29-36 8 p.

Research output

3 Citations (Scopus)

New nitrofurans amenable by isocyanide multicomponent chemistry are active against multidrug-resistant and poly-resistant Mycobacterium tuberculosis

Krasavin, M., Parchinsky, V., Kantin, G., Manicheva, O., Dogonadze, M., Vinogradova, T., Karge, B. & Brönstrup, M., 1 Jan 2017, In : Bioorganic and Medicinal Chemistry. 25, 6, p. 1867-1874 8 p.

Research output

12 Citations (Scopus)
2020
2017

Discovery of 4-amino-3-arylsulfoquinolines, a novel non-acetylenic chemotype of metabotropic glutamate 5 (mGlu5) receptor negative allosteric modulators

Galambos, J., Bielik, A., Wágner, G., Domány, G., Kóti, J., Béni, Z., Szigetvári, Á., Sánta, Z., Orgován, Z., Bobok, A., Kiss, B., Mikó-Bakk, M. L., Vastag, M., Sághy, K., Krasavin, M., Gál, K., Greiner, I., Szombathelyi, Z. & Keserű, G. M., 1 Jan 2017, In : European Journal of Medicinal Chemistry. 133, p. 240-254 15 p.

Research output

4 Citations (Scopus)

Continued SAR exploration of 1,2,4-thiadiazole-containing scaffolds in the design of free fatty acid receptor 1 (GPR40) agonists

Krasavin, M., Lukin, A., Bakholdina, A., Zhurilo, N., Onopchenko, O., Borysko, P., Zozulya, S., Moore, D. & Tikhonova, I. G., 1 Jan 2017, In : European Journal of Medicinal Chemistry. 140, p. 229-238 10 p.

Research output

5 Citations (Scopus)
2019
Open Access
6 Citations (Scopus)

Modern Trends of Organic Chemistry in Russian Universities

Konovalov, A. I., Antipin, I. S., Burilov, V. A., Madzhidov, T. I., Kurbangalieva, A. R., Nemtarev, A. V., Solovieva, S. E., Stoikov, I. I., Mamedov, V. A., Zakharova, L. Y., Gavrilova, E. L., Sinyashin, O. G., Balova, I. A., Vasilyev, A. V., Zenkevich, I. G., Krasavin, M. Y., Kuznetsov, M. A., Molchanov, A. P., Novikov, M. S., Nikolaev, V. A. & 59 others, Rodina, L. L., Khlebnikov, A. F., Beletskaya, I. P., Vatsadze, S. Z., Gromov, S. P., Zyk, N. V., Lebedev, A. T., Lemenovskii, D. A., Petrosyan, V. S., Nenaidenko, V. G., Negrebetskii, V. V., Baukov, Y. I., Shmigol’, T. A., Korlyukov, A. A., Tikhomirov, A. S., Shchekotikhin, A. E., Traven’, V. F., Voskresenskii, L. G., Zubkov, F. I., Golubchikov, O. A., Semeikin, A. S., Berezin, D. B., Stuzhin, P. A., Filimonov, V. D., Krasnokutskaya, E. A., Fedorov, A. Y., Nyuchev, A. V., Orlov, V. Y., Begunov, R. S., Rusakov, A. I., Kolobov, A. V., Kofanov, E. R., Fedotova, O. V., Egorova, A. Y., Charushin, V. N., Chupakhin, O. N., Klimochkin, Y. N., Osyanin, V. A., Reznikov, A. N., Fisyuk, A. S., Sagitullina, G. P., Aksenov, A. V., Aksenov, N. A., Grachev, M. K., Maslennikova, V. I., Koroteev, M. P., Brel’, A. K., Lisina, S. V., Medvedeva, S. M., Shikhaliev, K. S., Suboch, G. A., Tovbis, M. S., Mironovich, L. M., Ivanov, S. M., Kurbatov, S. V., Kletskii, M. E., Burov, O. N., Kobrakov, K. I. & Kuznetsov, D. N., 1 Feb 2018, In : Russian Journal of Organic Chemistry. 54, 2, p. 157-371 215 p.

Research output

43 Citations (Scopus)
2017

Discovery and Preclinical Characterization of 3-((4-(4-Chlorophenyl)-7-fluoroquinoline-3-yl)sulfonyl)benzonitrile, a Novel Non-acetylenic Metabotropic Glutamate Receptor 5 (mGluR5) Negative Allosteric Modulator for Psychiatric Indications

Galambos, J., Bielik, A., Krasavin, M., Orgován, Z., Domány, G., Nógrádi, K., Wágner, G., Balogh, G. T., Béni, Z., Kóti, J., Szakács, Z., Bobok, A., Kolok, S., Mikó-Bakk, M. L., Vastag, M., Sághy, K., Laszy, J., Halász, A. S., Balázs, O., Gál, K. & 3 others, Greiner, I., Szombathelyi, Z. & Keserű, G. M., 23 Mar 2017, In : Journal of Medicinal Chemistry. 60, 6, p. 2470-2484 15 p.

Research output

12 Citations (Scopus)
2018
19 Citations (Scopus)
2017
9 Citations (Scopus)
2020
1 Citation (Scopus)
2017
7 Citations (Scopus)
2020
1 Citation (Scopus)
2018
6 Citations (Scopus)
Open Access
2018

Discovery of polar spirocyclic orally bioavailable urea inhibitors of soluble epoxide hydrolase

Lukin, A., Kramer, J., Hartmann, M., Weizel, L., Hernandez-Olmos, V., Falahati, K., Burghardt, I., Kalinchenkova, N., Bagnyukova, D., Zhurilo, N., Rautio, J., Forsberg, M., Ihalainen, J., Auriola, S., Leppänen, J., Konstantinov, I., Pogoryelov, D., Proschak, E., Dar'in, D. & Krasavin, M., 1 Oct 2018, In : Bioorganic Chemistry. 80, p. 655-667 13 p.

Research output

8 Citations (Scopus)

Efficient Conversion of Tertiary Propargylamides into Imidazoles via Hydroamination-Cyclization

Safrygin, A., Krivosheyeva, E., Dar'in, D. & Krasavin, M., 1 Aug 2018, In : Synthesis (Germany). 50, 15, p. 3048-3058 11 p., ss-2018-z0257-op.

Research output

10 Citations (Scopus)
2017

Fluorescent (pyrazolyl acetoxime)Zn-II complexes: Synthetic, structural, and photophysical studies

Bolotin, D. S., Il'in, M. V., Kolesnikov, I. E., Suslonov, V. V., Novozhilov, Y., Ronzhina, O., Krasavin, M., Boyarskiy, V. P., Koen, R. & Roodt, A., 30 Jan 2017, In : Inorganica Chimica Acta. 455, p. 9-14 6 p.

Research output

3 Citations (Scopus)
2020
2017

Short Approach to Pyrrolopyrazino-, Pyrrolodiazepino-Isoindoles and their Benzo Analogues via the IMDAF Reaction

Zubkov, F. I., Orlova, D. N., Zaytsev, V. P., Voronov, A. A., Nikitina, E. V., Khrustalev, V. N., Novikov, R. A., Krasavin, M. & Varlamov, A. V., 2017, In : Current Organic Synthesis. 14, 5, p. 733-746 14 p.

Research output

2018

Conjugation of a 5-nitrofuran-2-oyl moiety to aminoalkylimidazoles produces non-toxic nitrofurans that are efficacious in vitro and in vivo against multidrug-resistant Mycobacterium tuberculosis

Krasavin, M., Lukin, A., Vedekhina, T., Manicheva, O., Dogonadze, M., Vinogradova, T., Zabolotnykh, N., Rogacheva, E., Kraeva, L. & Yablonsky, P., 5 Sep 2018, In : European Journal of Medicinal Chemistry. 157, p. 1115-1126 12 p.

Research output

2 Citations (Scopus)
2016
7 Citations (Scopus)

Gram-scale synthesis of a novel core building block for the new GPR40 agonist design

Lukin, A., Bagnyukova, D., Zhurilo, N. & Krasavin, M., 1 Aug 2016, In : Letters in Organic Chemistry. 13, 7, p. 491-495 5 p.

Research output

2 Citations (Scopus)

New antimycobacterial leads from multicomponent hydrazino-ugi reaction

Lakontseva, E., Karapetian, R. & Krasavin, M., 1 Mar 2016, In : Medicinal Chemistry. 12, 2, p. 191-199 9 p.

Research output

2 Citations (Scopus)
2020

Exploring bulky natural and natural-like periphery in the design of p-(benzyloxy)phenylpropionic acid agonists of free fatty acid receptor 1 (GPR40)

Kuranov, S. O., Luzina, O. A., Onopchenko, O., Pishel, I., Zozulya, S., Gureev, M., Salakhutdinov, N. F. & Krasavin, M., Jun 2020, In : Bioorganic Chemistry. 99, 103830.

Research output

2016
19 Citations (Scopus)
2017
7 Citations (Scopus)