Find Research outputs — Saint Petersburg State University

2016

Double tandem cyclization of 4-(1-acyl-2,2-diaminovinyl)-6-arylpyrimidine-5-carbonitriles. Synthesis of novel peri-annulated azines.

Putintseva, M. N., Bakulina, O. Y., Ivanov, A. Y., Lobanov, P. S., Nikolskaya, S. K., Kolesnikov, I. E. & Dar’in, D. V., 2016, In : Tetrahedron Letters. 57, p. 5192-5196

Research output

1 Citation (Scopus)

2014

New transformations of 2-methylsulfanyl-4,6-dichloropyrimidine-5‑carbaldehyde involving enamines: synthesis of condensed azines

Bakulina, O. Y., Ivanov, A. Y., Dar'In, D. V. & Lobanov, P. S., 2014, In : Mendeleev Communications. 3, p. 163-164

Research output

6 Citations (Scopus)

2018

A General Way to Construct Arene-Fused Seven-Membered Nitrogen Heterocycles

Bakulina, O., Chizhova, M., Dar'in, D. & Krasavin, M., 23 Jan 2018, In : European Journal of Organic Chemistry. 2018, 3, p. 362-371 10 p.

Research output

11 Citations (Scopus)

2019

Facile access to Fe(III)-complexing cyclic hydroxamic acids in a three-component format

Chupakhin, E., Bakulina, O., Dar’in, D. & Krasavin, M., 1 Mar 2019, In : Molecules. 24, 5, 15 p., 864.

Research output

Open Access

3 Citations (Scopus)

2020

Two annulated azaheterocyclic cores readily available from a single tetrahydroisoquinolonic Castagnoli–Cushman precursor

Karchuganova, E., Bakulina, O., Dar’in, D. & Krasavin, M., May 2020, In : Molecules. 25, 9, 2049.

Research output

Open Access

Synthesis of spirocyclic tetrahydroisoquinolines (spiroTHIQs) via the Castagnoli-Cushman reaction

Safrygin, A., Dar'in, D., Bakulina, O. & Krasavin, M., 31 Aug 2020, In : Tetrahedron Letters. 152408.

Research output

Three-Component Reaction of Homophthalic Anhydride with Carbonyl Compounds and Ammonium Acetate: New Developments

Safrygin, A., Bakulina, O., Dar'In, D. & Krasavin, M., 4 Aug 2020, In : Synthesis (Germany). 52, 15, p. 2190-2195 6 p.

Research output

1 Citation (Scopus)

From Rare Reagents to Rare Products: Regiospecific Silver-Catalyzed [3+2] Cycloaddition of Aryl-, Alkyl- and Aminosulfonyl Diazomethanes with Arenediazonium Tosylates

Levashova, E., Bakulina, O., Dar'in, D., Bubyrev, A., Chuprun, S. & Krasavin, M., 7 Jul 2020, In : European Journal of Organic Chemistry. 5 p.

Research output

1 Citation (Scopus)

2016

Indoline-Based Constrained Peptidomimetic Motifs Obtained via the Joullié–Ugi Reaction of Indolenines.

Golubev, P., Bakulina, O., Dar'in, D. & Krasavin, M., 2016, In : European Journal of Organic Chemistry. p. 3969-3976

Research output

9 Citations (Scopus)

2019

The use of ∝-diazo-γ-butyrolactone in the Büchner-Curtius-Schlotterbeck reaction of cyclic ketones: A facile entry into spirocyclic scaffolds

Shershnev, I., Dar'in, D. V., Chuprun, S. S., Kantin, G. P., Bakulina, O. Y. & Krasavin, M., 4 Jul 2019, In : Tetrahedron Letters. 60, 27, p. 1800-1802 3 p.

Research output

7 Citations (Scopus)

2020

Dialkyl diazomalonates in transition-metal-free, thermally promoted, diastereoselective wolff β-lactam synthesis

Synofzik, J., Bakulina, O., Dar'in, D., Kantin, G. & Krasavin, M., 12 Aug 2020, In : Synlett. 31, 13, p. 1273-1276 4 p.

Research output

1 Citation (Scopus)

Catalyst-Free Synthesis of Diastereomerically Pure 3-Sulfonyl azetidin-2-ones via Microwave-Assisted Tandem Wolff Rearrangement-Staudinger Cycloaddition

Synofzik, J., Bakulina, O., Balabas, O., Dar'In, D. & Krasavin, M., 21 Jul 2020, In : Synthesis (Germany).

Research output

Dual use of propargylamine building blocks in the construction of polyheterocyclic scaffolds

Bakholdina, A., Lukin, A., Bakulina, O., Guranova, N. & Krasavin, M., 23 Apr 2020, In : Tetrahedron Letters. 151970.

Research output

2015

Facile synthesis of pyrido[2,3-d]pyrimidines via cyclocondensation of 4,6-dichloro-2-methylsulfanylpyrimidine-5-carbaldehyde with β-substituted β-aminoacrylic esters

Chizhova, M. E., Bakulina, O. Y., Ivanov, A. Y., Lobanov, P. S. & Dar'in, D. V., 2015, In : Tetrahedron. 71, 36, p. 6196-6203 8 p.

Research output

5 Citations (Scopus)

2013

Reaction of ethyl 3,3-diaminoacrylate with pyrimidine series o-chloro ketones. Synthesis of pyrido[4,3-d]pyrimidines and 6H-1,3,6,7-tetra-azaphenalenes

Bakulina, O. Y., Igumnova, E. M., Dar'In, D. V. & Lobanov, P. S., 2013, In : Chemistry of Heterocyclic Compounds. 49, 3, p. 466-471

Research output

6 Citations (Scopus)

2018

Synthesis of Water-Soluble Blue-Emissive Tricyclic 2-Aminopyridinium Salts by Three-Component Coupling-(3+3)-Anellation

Bakulina, O., Merkt, F. K., Knedel, T. O., Janiak, C. & Müller, T. J. J., 21 Dec 2018, In : Angewandte Chemie - International Edition. 57, 52, p. 17240-17244 5 p.

Research output

5 Citations (Scopus)

2015

New Heterocyclic Product Space for the Castagnoli-Cushman Three-Component Reaction

Dar'In, D., Bakulina, O., Chizhova, M. & Krasavin, M., 2015, In : Organic Letters. p. 3930-3933

Research output

47 Citations (Scopus)

2020

Straightforward Route to gamma-Sultams via Novel Tandem S-N/Michael Addition

Klochkova, A., Bubyrev, A., Dar'in, D., Bakulina, O., Krasavin, M. & Sokolov, V., 29 Dec 2020, In : Synthesis. 10 p.

Research output

2019

Rh(II)-Catalyzed spirocyclization of α-diazo homophthalimides with cyclic ethers

Guranova, N. I., Dar’in, D., Kantin, G., Novikov, A. S., Bakulina, O. & Krasavin, M., 5 Apr 2019, In : The Journal of organic chemistry. 84, 7, p. 4534-4542 9 p.

Research output

9 Citations (Scopus)

Fused vs. spiro: Kinetic, not thermodynamic preference may direct the reaction of alpha-carbonyl oxonium ylides

Guranova, N. I., Dar'in, D., Kantin, G., Novikov, A. S., Bakulina, O. & Krasavin, M., 13 Jun 2019, In : Tetrahedron Letters. 60, 24, p. 1582-1586 5 p.

Research output

1 Citation (Scopus)

2018

Concise synthesis of 2-N-hydroxy-3,4-dihydroisoquinol-2-one: A bacterial siderophore and human 5-lipooxygenase inhibitor

Tutov, A., Bakulina, O., Dar'in, D. & Krasavin, M., 11 Apr 2018, In : Tetrahedron Letters. 59, 15, p. 1511-1512 2 p.

Research output

5 Citations (Scopus)

2019

Three-Component Castagnoli-Cushman Reaction of 3-Arylglutaconic Acids with Aromatic Aldehydes and Amines Delivers Rare 4,6-Diaryl-1,6-dihydropyridin-2(3 H)-ones

Firsov, A., Chupakhin, E., Dar'In, D., Bakulina, O. & Krasavin, M., 15 Mar 2019, In : Organic Letters. 21, 6, p. 1637-1640

Research output

3 Citations (Scopus)

Flexible Entry into 3-Arylpent-2-enedioic Acids via Heck-Matsuda Arylation of Dimethyl Glutaconate with Arenediazonium Tosylates

Dar'In, D., Kantin, G., Bakulina, O., Žalubovskis, R. & Krasavin, M., May 2019, In : Synthesis (Germany). 51, 10, p. 2230-2236 7 p.

Research output

Open Access

3 Citations (Scopus)

2020

Facile One-Pot Access to α-Diazo-β-ketosulfones from Sulfonyl Chlorides and α-Haloketones

Dar'In, D., Kantin, G., Bakulina, O. & Krasavin, M., 4 Aug 2020, In : Synthesis (Germany). 52, 15, p. 2259-2266 8 p.

Research output

3 Citations (Scopus)

2019

Modular Assembly of Tunable Fluorescent Chemosensors Selective for Pb²⁺ and Cu²⁺ Metal Ions via the Multicomponent Castagnoli-Cushman Reaction

Bakulina, O., Rashevskii, A., Dar'in, D., Halder, S., Khagar, P. & Krasavin, M., 31 May 2019, In : ChemistrySelect. 4, 20, p. 6066-6073

Research output

1 Citation (Scopus)

2018

Design, in silico prioritization and biological profiling of apoptosis-inducing lactams amenable by the Castagnoli-Cushman reaction

Krasavin, M., Gureyev, M. A., Dar'in, D., Bakulina, O., Chizhova, M., Lepikhina, A., Novikova, D., Grigoreva, T., Ivanov, G., Zhumagalieva, A., Garabadzhiu, A. V. & Tribulovich, V. G., 15 May 2018, In : Bioorganic and Medicinal Chemistry. 26, 9, p. 2651-2673 23 p.

Research output

5 Citations (Scopus)

2019

1,1′-Carbonyldiimidazole as a cyclodehydrating agent for the Castagnoli–Cushman reaction of dicarboxylic acids and imines

Chupakhin, E. G., Bakulina, O. Y., Dar'in, D. V. & Krasavin, M., 1 May 2019, In : Mendeleev Communications . 29, 3, p. 292-293

Research output

2 Citations (Scopus)

2018

Mixed carboxylic-sulfonic anhydride in reaction with imines: A straightforward route to water-soluble β-lactams via a Staudinger-type reaction

Bakulina, O., Dar'in, D. & Krasavin, M., 1 Jan 2018, In : Organic and Biomolecular Chemistry. 16, 21, p. 3989-3998 10 p.

Research output

3 Citations (Scopus)

2014

Synthesis of novel peri-fused heterocyclic systems - pyrimido[4,5,6-de][1,8]naphthyridines, based on interaction of 4,6-dichloro-2-methylthiopyrimidine-5-carbaldehyde with geminal enediamines

Bakulina, O. Y., Ivanov, A. Y., Lobanov, P. S. & Dar'In, D. V., 2014, In : Tetrahedron. 70, 43, p. 7900-7905

Research output

6 Citations (Scopus)

2020

The Future of Scientific Leadership is Interdisciplinary: The 2019 CAS Future Leaders Share Their Vision

V. Milić, J., Ehnbom, A., Garedew, M., Vincent-Ruz, P., Schloemer, T. H., Hodgson, G. K., Oakley, M. S., Sasaki, K., Chander, S., Légaré, M. A., Callmann, C. E., Bismillah, A. N., van Osch, D. J. G. P., Sanchez, V., Boase, N. R. B., Mambwe, D., Coley, C. W., Deng, Y., Betz, K. N., Sanjosé-Orduna, J. & 9 others, Natoli, S., Zhang, L., Bakulina, O., Fereyduni, E., Hilario-Martínez, J. C., Busta, L., Hunter, A., Park, Y. & Zadeh, F. H., 25 Sep 2020, In : iScience. 23, 9, 101442.

Research output

Open Access

2016

The rare cis-configured trisubstituted lactam products obtained by the Castagnoli-Cushman reaction in N,N-dimethylformamide.

Dar'in, D., Bakulina, O., Nikolskaya, S., Gluzdikov, I. & Krasavin, M., 2016, In : RSC Advances. p. 49411-49415

Research output

16 Citations (Scopus)

2020

One-pot preparation of methyl 2-diazo-3-oxopropionates comprising an aqueous ‘sulfonyl-azide-free’ (SAFE) diazo transfer step

Zhmurov, P. A., Dar'in, D. V., Bakulina, O. Y. & Krasavin, M., 2020, In : Mendeleev Communications . 30, 3, p. 311-312 2 p.

Research output

2016

New Dicarboxylic Acid Anhydride for Ambient-Temperature Castagnoli-Cushman Reactions

Chizhova, M., Bakulina, O., Dar'in, D. & Krasavin, M., 2016, In : ChemistrySelect. 1, 17, p. 5487-5492

Research output

4 Citations (Scopus)

2020

Spirocyclizations Involving Oxonium Ylides Derived from Cyclic α-Diazocarbonyl Compounds: An Entry into 6-Oxa-2-azaspiro[4.5]decane Scaffold

Dar'in, D., Kantin, G., Bakulina, O., Inyutina, A., Chupakhin, E. & Krasavin, M., 2020, In : Journal of Organic Chemistry. 85, 23, p. 15586–15599

Research output

1 Citation (Scopus)

Further Insight into the Castagnoli-Cushman-type Synthesis of 1,4,6-Trisubstituted 1,6-Dihydropyridin-2-(3 H)-ones from 3-Arylglutaconic Acid Anhydrides

Firsov, A., Bakulina, O., Dar'in, D., Guranova, N. & Krasavin, M., 1 Jan 2020, In : Journal of Organic Chemistry.

Research output

When periphery matters: Enhanced reactivity of 8-oxa-1,4-dithiaspiro[4.5]decane-7,9-dione and 9-oxa-1,5-dithiaspiro[5.5]undecane-8,10-dione in the Castagnoli-Cushman reaction with imines

Rashevskii, A., Bakulina, O., Novikov, M. S., Dar'in, D. & Krasavin, M., 2020, (Accepted/In press) In : Tetrahedron Letters. 61, 52, 152658.

Research output

2016

The first solvent-free synthesis of privileged γ- and δ-lactams via the Castagnoli–Cushman reaction.

Lepikhina, A., Bakulina, O., Dar'in, D. & Krasavin, M., 2016, In : RSC Advances. 6, p. 83808-83813

Research output

15 Citations (Scopus)

2019

Design, synthesis, and biological evaluation of novel derivatives of dithiodiglycolic acid prepared via oxidative coupling of thiols

Bakulina, O., Bannykh, A., Jovanović, M., Domračeva, I., Podolski-Renić, A., Žalubovskis, R., Pešić, M., Dar’in, D. & Krasavin, M., 1 Jan 2019, In : Journal of Enzyme Inhibition and Medicinal Chemistry. 34, 1, p. 665-671 7 p.

Research output

3 Citations (Scopus)

Hydroxylamine as an ammonia equivalent: access to NH-tetrahydroisoquinolonic derivatives from aldoximes by the Castagnoli–Cushman reaction followed by reduction

Bannykh, A. V., Bakulina, O. Y., Dar'in, D. V. & Krasavin, M., 1 May 2019, In : Mendeleev Communications . 29, 3, p. 337-338

Research output

1 Citation (Scopus)

α-Acyl-α-diazoacetates in Transition-Metal-Free β-Lactam Synthesis

Synofzik, J., Dar'In, D., Novikov, M. S., Kantin, G., Bakulina, O. & Krasavin, M., 20 Sep 2019, In : Journal of Organic Chemistry. 84, 18, p. 12101-12110

Research output

6 Citations (Scopus)

2020

Mutually isomeric 2-and 4-(3-nitro-1,2,4-triazol-1yl)pyrimidines inspired by an antimycobacterial screening hit: Synthesis and biological activity against the eskape panel of pathogens

Chuprun, S., Dar’in, D., Rogacheva, E., Kraeva, L., Levin, O., Manicheva, O., Dogonadze, M., Vinogradova, T., Bakulina, O. & Krasavin, M., 1 Oct 2020, In : Antibiotics. 9, 10, p. 1-21 21 p., 666.

Research output

Open Access

2019

Aryl-Aryl Coupling of Salicylic Aldehydes through Oxidative CH-activation in Nickel Salen Derivatives

Yankin, A. N., Lukyanov, D. A., Beletskii, E. V., Bakulina, O. Y., Vlasov, P. S. & Levin, O. V., 12 Aug 2019, In : ChemistrySelect. 4, 30, p. 8886-8890

Research output

2 Citations (Scopus)

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