Find Research outputs — Saint Petersburg State University

2016

Double tandem cyclization of 4-(1-acyl-2,2-diaminovinyl)-6-arylpyrimidine-5-carbonitriles. Synthesis of novel peri-annulated azines.

Putintseva, M. N., Bakulina, O. Y., Ivanov, A. Y., Lobanov, P. S., Nikolskaya, S. K., Kolesnikov, I. E. & Dar’in, D. V., 2016, In : Tetrahedron Letters. 57, p. 5192-5196

Research output

1 Citation (Scopus)

2014

New transformations of 2-methylsulfanyl-4,6-dichloropyrimidine-5‑carbaldehyde involving enamines: synthesis of condensed azines

Bakulina, O. Y., Ivanov, A. Y., Dar'In, D. V. & Lobanov, P. S., 2014, In : Mendeleev Communications. 3, p. 163-164

Research output

6 Citations (Scopus)

2017

Spontaneous formation of tricyclic lactones following the Castagnoli–Cushman reaction

Usmanova, L., Bakulina, O., Dar’in, D. & Krasavin, M., 1 Apr 2017, In : Chemistry of Heterocyclic Compounds. 53, 4, p. 474-479 6 p.

Research output

2018

A General Way to Construct Arene-Fused Seven-Membered Nitrogen Heterocycles

Bakulina, O., Chizhova, M., Dar'in, D. & Krasavin, M., 23 Jan 2018, In : European Journal of Organic Chemistry. 2018, 3, p. 362-371 10 p.

Research output

11 Citations (Scopus)

2017

Cyclic Hydroxamic Acid Analogues of Bacterial Siderophores as Iron-Complexing Agents prepared through the Castagnoli–Cushman Reaction of Unprotected Oximes

Bakulina, O., Bannykh, A., Dar'in, D. & Krasavin, M., 14 Dec 2017, In : Chemistry - A European Journal. 23, 70, p. 17667-17673 7 p.

Research output

8 Citations (Scopus)

2020

Two annulated azaheterocyclic cores readily available from a single tetrahydroisoquinolonic Castagnoli–Cushman precursor

Karchuganova, E., Bakulina, O., Dar’in, D. & Krasavin, M., May 2020, In : Molecules. 25, 9, 2049.

Research output

Open Access

Synthesis of spirocyclic tetrahydroisoquinolines (spiroTHIQs) via the Castagnoli-Cushman reaction

Safrygin, A., Dar'in, D., Bakulina, O. & Krasavin, M., 31 Aug 2020, In : Tetrahedron Letters. 152408.

Research output

Three-Component Reaction of Homophthalic Anhydride with Carbonyl Compounds and Ammonium Acetate: New Developments

Safrygin, A., Bakulina, O., Dar'In, D. & Krasavin, M., 4 Aug 2020, In : Synthesis (Germany). 52, 15, p. 2190-2195 6 p.

Research output

1 Citation (Scopus)

From Rare Reagents to Rare Products: Regiospecific Silver-Catalyzed [3+2] Cycloaddition of Aryl-, Alkyl- and Aminosulfonyl Diazomethanes with Arenediazonium Tosylates

Levashova, E., Bakulina, O., Dar'in, D., Bubyrev, A., Chuprun, S. & Krasavin, M., 7 Jul 2020, In : European Journal of Organic Chemistry. 5 p.

Research output

1 Citation (Scopus)

2016

Indoline-Based Constrained Peptidomimetic Motifs Obtained via the Joullié–Ugi Reaction of Indolenines.

Golubev, P., Bakulina, O., Dar'in, D. & Krasavin, M., 2016, In : European Journal of Organic Chemistry. p. 3969-3976

Research output

9 Citations (Scopus)

2017

o-Phenylenediacetic Acid Anhydride in the Castagnoli–Cushman Reaction: Extending the Product Space to ε-Lactams

Bakulina, O., Dar’in, D. & Krasavin, M., 2017, In : Synlett. 28, 10, p. 1165-1169

Research output

13 Citations (Scopus)

2020

Dialkyl diazomalonates in transition-metal-free, thermally promoted, diastereoselective wolff β-lactam synthesis

Synofzik, J., Bakulina, O., Dar'in, D., Kantin, G. & Krasavin, M., 12 Aug 2020, In : Synlett. 31, 13, p. 1273-1276 4 p.

Research output

1 Citation (Scopus)

Catalyst-Free Synthesis of Diastereomerically Pure 3-Sulfonyl azetidin-2-ones via Microwave-Assisted Tandem Wolff Rearrangement-Staudinger Cycloaddition

Synofzik, J., Bakulina, O., Balabas, O., Dar'In, D. & Krasavin, M., 21 Jul 2020, In : Synthesis (Germany).

Research output

Dual use of propargylamine building blocks in the construction of polyheterocyclic scaffolds

Bakholdina, A., Lukin, A., Bakulina, O., Guranova, N. & Krasavin, M., 23 Apr 2020, In : Tetrahedron Letters. 151970.

Research output

2015

Facile synthesis of pyrido[2,3-d]pyrimidines via cyclocondensation of 4,6-dichloro-2-methylsulfanylpyrimidine-5-carbaldehyde with β-substituted β-aminoacrylic esters

Chizhova, M. E., Bakulina, O. Y., Ivanov, A. Y., Lobanov, P. S. & Dar'in, D. V., 2015, In : Tetrahedron. 71, 36, p. 6196-6203 8 p.

Research output

5 Citations (Scopus)

2013

Reaction of ethyl 3,3-diaminoacrylate with pyrimidine series o-chloro ketones. Synthesis of pyrido[4,3-d]pyrimidines and 6H-1,3,6,7-tetra-azaphenalenes

Bakulina, O. Y., Igumnova, E. M., Dar'In, D. V. & Lobanov, P. S., 2013, In : Chemistry of Heterocyclic Compounds. 49, 3, p. 466-471

Research output

6 Citations (Scopus)

2018

Synthesis of Water-Soluble Blue-Emissive Tricyclic 2-Aminopyridinium Salts by Three-Component Coupling-(3+3)-Anellation

Bakulina, O., Merkt, F. K., Knedel, T. O., Janiak, C. & Müller, T. J. J., 21 Dec 2018, In : Angewandte Chemie - International Edition. 57, 52, p. 17240-17244 5 p.

Research output

5 Citations (Scopus)

2015

New Heterocyclic Product Space for the Castagnoli-Cushman Three-Component Reaction

Dar'In, D., Bakulina, O., Chizhova, M. & Krasavin, M., 2015, In : Organic Letters. p. 3930-3933

Research output

47 Citations (Scopus)

2020

Straightforward Route to gamma-Sultams via Novel Tandem S-N/Michael Addition

Klochkova, A., Bubyrev, A., Dar'in, D., Bakulina, O., Krasavin, M. & Sokolov, V., 29 Dec 2020, In : Synthesis. 10 p.

Research output

2018

Concise synthesis of 2-N-hydroxy-3,4-dihydroisoquinol-2-one: A bacterial siderophore and human 5-lipooxygenase inhibitor

Tutov, A., Bakulina, O., Dar'in, D. & Krasavin, M., 11 Apr 2018, In : Tetrahedron Letters. 59, 15, p. 1511-1512 2 p.

Research output

5 Citations (Scopus)

2017

Skeletal Diversity in Combinatorial Fashion: A New Format for the Castagnoli-Cushman Reaction

Lepikhina, A., Dar'In, D., Bakulina, O., Chupakhin, E. & Krasavin, M., 13 Nov 2017, In : ACS Combinatorial Science. 19, 11, p. 702-707 6 p.

Research output

14 Citations (Scopus)

2020

Facile One-Pot Access to α-Diazo-β-ketosulfones from Sulfonyl Chlorides and α-Haloketones

Dar'In, D., Kantin, G., Bakulina, O. & Krasavin, M., 4 Aug 2020, In : Synthesis (Germany). 52, 15, p. 2259-2266 8 p.

Research output

3 Citations (Scopus)

2018

Design, in silico prioritization and biological profiling of apoptosis-inducing lactams amenable by the Castagnoli-Cushman reaction

Krasavin, M., Gureyev, M. A., Dar'in, D., Bakulina, O., Chizhova, M., Lepikhina, A., Novikova, D., Grigoreva, T., Ivanov, G., Zhumagalieva, A., Garabadzhiu, A. V. & Tribulovich, V. G., 15 May 2018, In : Bioorganic and Medicinal Chemistry. 26, 9, p. 2651-2673 23 p.

Research output

5 Citations (Scopus)

Mixed carboxylic-sulfonic anhydride in reaction with imines: A straightforward route to water-soluble β-lactams via a Staudinger-type reaction

Bakulina, O., Dar'in, D. & Krasavin, M., 1 Jan 2018, In : Organic and Biomolecular Chemistry. 16, 21, p. 3989-3998 10 p.

Research output

3 Citations (Scopus)

2014

Synthesis of novel peri-fused heterocyclic systems - pyrimido[4,5,6-de][1,8]naphthyridines, based on interaction of 4,6-dichloro-2-methylthiopyrimidine-5-carbaldehyde with geminal enediamines

Bakulina, O. Y., Ivanov, A. Y., Lobanov, P. S. & Dar'In, D. V., 2014, In : Tetrahedron. 70, 43, p. 7900-7905

Research output

6 Citations (Scopus)

2020

The Future of Scientific Leadership is Interdisciplinary: The 2019 CAS Future Leaders Share Their Vision

V. Milić, J., Ehnbom, A., Garedew, M., Vincent-Ruz, P., Schloemer, T. H., Hodgson, G. K., Oakley, M. S., Sasaki, K., Chander, S., Légaré, M. A., Callmann, C. E., Bismillah, A. N., van Osch, D. J. G. P., Sanchez, V., Boase, N. R. B., Mambwe, D., Coley, C. W., Deng, Y., Betz, K. N., Sanjosé-Orduna, J. & 9 others, Natoli, S., Zhang, L., Bakulina, O., Fereyduni, E., Hilario-Martínez, J. C., Busta, L., Hunter, A., Park, Y. & Zadeh, F. H., 25 Sep 2020, In : iScience. 23, 9, 101442.

Research output

Open Access

2016

The rare cis-configured trisubstituted lactam products obtained by the Castagnoli-Cushman reaction in N,N-dimethylformamide.

Dar'in, D., Bakulina, O., Nikolskaya, S., Gluzdikov, I. & Krasavin, M., 2016, In : RSC Advances. p. 49411-49415

Research output

16 Citations (Scopus)

2020

One-pot preparation of methyl 2-diazo-3-oxopropionates comprising an aqueous ‘sulfonyl-azide-free’ (SAFE) diazo transfer step

Zhmurov, P. A., Dar'in, D. V., Bakulina, O. Y. & Krasavin, M., 2020, In : Mendeleev Communications . 30, 3, p. 311-312 2 p.

Research output

2016

New Dicarboxylic Acid Anhydride for Ambient-Temperature Castagnoli-Cushman Reactions

Chizhova, M., Bakulina, O., Dar'in, D. & Krasavin, M., 2016, In : ChemistrySelect. 1, 17, p. 5487-5492

Research output

4 Citations (Scopus)

2020

Spirocyclizations Involving Oxonium Ylides Derived from Cyclic α-Diazocarbonyl Compounds: An Entry into 6-Oxa-2-azaspiro[4.5]decane Scaffold

Dar'in, D., Kantin, G., Bakulina, O., Inyutina, A., Chupakhin, E. & Krasavin, M., 2020, In : Journal of Organic Chemistry. 85, 23, p. 15586–15599

Research output

1 Citation (Scopus)

Further Insight into the Castagnoli-Cushman-type Synthesis of 1,4,6-Trisubstituted 1,6-Dihydropyridin-2-(3 H)-ones from 3-Arylglutaconic Acid Anhydrides

Firsov, A., Bakulina, O., Dar'in, D., Guranova, N. & Krasavin, M., 1 Jan 2020, In : Journal of Organic Chemistry.

Research output

When periphery matters: Enhanced reactivity of 8-oxa-1,4-dithiaspiro[4.5]decane-7,9-dione and 9-oxa-1,5-dithiaspiro[5.5]undecane-8,10-dione in the Castagnoli-Cushman reaction with imines

Rashevskii, A., Bakulina, O., Novikov, M. S., Dar'in, D. & Krasavin, M., 2020, (Accepted/In press) In : Tetrahedron Letters. 61, 52, 152658.

Research output

2017

A speedy route to sterically encumbered, benzene-fused derivatives of privileged, naturally occurring hexahydropyrrolo[1,2-b]isoquinoline

Bakulina, O., Ivanov, A., Suslonov, V., Darin, D. & Krasavin, M., 18 Jul 2017, In : Beilstein Journal of Organic Chemistry. 13, p. 1413-1424 12 p.

Research output

10 Citations (Scopus)

2016

The first solvent-free synthesis of privileged γ- and δ-lactams via the Castagnoli–Cushman reaction.

Lepikhina, A., Bakulina, O., Dar'in, D. & Krasavin, M., 2016, In : RSC Advances. 6, p. 83808-83813

Research output

15 Citations (Scopus)

2020

Mutually isomeric 2-and 4-(3-nitro-1,2,4-triazol-1yl)pyrimidines inspired by an antimycobacterial screening hit: Synthesis and biological activity against the eskape panel of pathogens

Chuprun, S., Dar’in, D., Rogacheva, E., Kraeva, L., Levin, O., Manicheva, O., Dogonadze, M., Vinogradova, T., Bakulina, O. & Krasavin, M., 1 Oct 2020, In : Antibiotics. 9, 10, p. 1-21 21 p., 666.

Research output

Open Access

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