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  1. 2019

  2. Pyridazinone-substituted benzenesulfonamides display potent inhibition of membrane-bound human carbonic anhydrase IX and promising antiproliferative activity against cancer cell lines

    Krasavin, M., Shetnev, A., Baykov, S., Kalinin, S., Nocentini, A., Sharoyko, V., Poli, G., Tuccinardi, T., Korsakov, M., Tennikova, T. B. & Supuran, C. T., 15 Apr 2019, In: European Journal of Medicinal Chemistry. 168, p. 301-314 14 p.

    Research output: Contribution to journal › Article › peer-review

  3. 1,2,4-Oxadiazole/2-Imidazoline Hybrids: Multi-target-directed Compounds for the Treatment of Infectious Diseases and Cancer

    Shetnev, A., Baykov, S., Kalinin, S., Belova, A., Sharoyko, V., Rozhkov, A., Zelenkov, L., Tarasenko, M., Sadykov, E., Korsakov, M. & Krasavin, M., 1 Apr 2019, In: International Journal of Molecular Sciences. 20, 7, p. 1699 10 p., 1699.

    Research output: Contribution to journal › Article › peer-review

  4. Continued exploration of 1,2,4-oxadiazole periphery for carbonic anhydrase-targeting primary arene sulfonamides: Discovery of subnanomolar inhibitors of membrane-bound hCA IX isoform that selectively kill cancer cells in hypoxic environment

    Krasavin, M., Shetnev, A., Sharonova, T., Baykov, S., Kalinin, S., Nocentini, A., Sharoyko, V., Poli, G., Tuccinardi, T., Presnukhina, S., Tennikova, T. B. & Supuran, C. T., 15 Feb 2019, In: European Journal of Medicinal Chemistry. 164, p. 92-105

    Research output: Contribution to journal › Article › peer-review

  5. 2018

  6. Heterocyclic periphery in the design of carbonic anhydrase inhibitors: 1,2,4-Oxadiazol-5-yl benzenesulfonamides as potent and selective inhibitors of cytosolic hCA II and membrane-bound hCA IX isoforms

    Krasavin, M., Shetnev, A., Sharonova, T., Baykov, S., Tuccinardi, T., Kalinin, S., Angeli, A. & Supuran, C. T., 1 Feb 2018, In: Bioorganic Chemistry. 76, p. 88-97 10 p.

    Research output: Contribution to journal › Article › peer-review

  7. Unprotected primary sulfonamide group facilitates ring-forming cascade en route to polycyclic [1,4]oxazepine-based carbonic anhydrase inhibitors

    Sapegin, A., Kalinin, S., Angeli, A., Supuran, C. T. & Krasavin, M., 1 Feb 2018, In: Bioorganic Chemistry. 76, p. 140-146 7 p.

    Research output: Contribution to journal › Article › peer-review

  8. 2017

  9. Lucky Switcheroo: Dramatic Potency and Selectivity Improvement of Imidazoline Inhibitors of Human Carbonic Anhydrase VII

    Kalinin, S., Kopylov, S., Tuccinardi, T., Sapegin, A., Dar'In, D., Angeli, A., Supuran, C. T. & Krasavin, M., 12 Oct 2017, In: ACS Medicinal Chemistry Letters. 8, 10, p. 1105-1109 5 p.

    Research output: Contribution to journal › Article › peer-review

  10. Human carbonic anhydrase inhibitory profile of mono- and bis-sulfonamides synthesized via a direct sulfochlorination of 3- and 4-(hetero)arylisoxazol-5-amine scaffolds

    Krasavin, M., Korsakov, M., Zvonaryova, Z., Semyonychev, E., Tuccinardi, T., Kalinin, S., Tanç, M. & Supuran, C. T., 1 Jan 2017, In: Bioorganic and Medicinal Chemistry. 25, 6, p. 1914-1925 12 p.

    Research output: Contribution to journal › Article › peer-review

  11. Primary mono- and bis-sulfonamides obtained via regiospecific sulfochlorination of N-arylpyrazoles: inhibition profile against a panel of human carbonic anhydrases

    Krasavin, M., Korsakov, M., Ronzhina, O., Tuccinardi, T., Kalinin, S., Tanç, M. & Supuran, C. T., 1 Jan 2017, In: Journal of Enzyme Inhibition and Medicinal Chemistry. 32, 1, p. 920-934 15 p.

    Research output: Contribution to journal › Article › peer-review

  12. The first one-pot ambient-temperature synthesis of 1,2,4-oxadiazoles from amidoximes and carboxylic acid esters

    Baykov, S., Sharonova, T., Shetnev, A., Rozhkov, S., Kalinin, S. & Smirnov, A. V., 1 Jan 2017, In: Tetrahedron. 73, 7, p. 945-951 7 p.

    Research output: Contribution to journal › Article › peer-review

  13. 2016

  14. Isoform-selective inhibitory profile of 2-imidazoline-substituted benzenesulfonamides against a panel of human carbonic anhydrases.

    Supuran, C. T., Kalinin, S., Tanç, M., Sarnpitak, P., Mujumdar, P., Poulsen, SA. & Krasavin, M., 2016, In: Journal of Enzyme Inhibition and Medicinal Chemistry. 31 (Suppl. 1), p. 197-202

    Research output: Contribution to journal › Article › peer-review

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